Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0005576 | cellular_component | extracellular region |
A | 0006952 | biological_process | defense response |
A | 0008200 | molecular_function | ion channel inhibitor activity |
A | 0017080 | molecular_function | sodium channel regulator activity |
A | 0019871 | molecular_function | sodium channel inhibitor activity |
A | 0035821 | biological_process | modulation of process of another organism |
A | 0090729 | molecular_function | toxin activity |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE MPD A 101 |
Chain | Residue |
A | TRP39 |
A | ILE40 |
A | GLY41 |
A | GLU55 |
A | MPD102 |
A | HOH221 |
site_id | AC2 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE MPD A 102 |
Chain | Residue |
A | TRP39 |
A | ILE40 |
A | MPD101 |
A | MPD103 |
A | TYR6 |
A | LYS29 |
A | ASN30 |
site_id | AC3 |
Number of Residues | 9 |
Details | BINDING SITE FOR RESIDUE MPD A 103 |
Chain | Residue |
A | ILE7 |
A | ALA8 |
A | ASP9 |
A | ASP10 |
A | ASP10 |
A | TYR15 |
A | ASN30 |
A | VAL56 |
A | MPD102 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | SITE: Important for toxin potency but not for selectivity for individual Nav channel subtype (Nav1.6/SCN8A and Nav1.7/SCN9A) => ECO:0000269|PubMed:23527544 |
Chain | Residue | Details |
A | ARG65 | |