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4F49

2.25A resolution structure of Transmissible Gastroenteritis Virus Protease containing a covalently bound Dipeptidyl Inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
B0008233molecular_functionpeptidase activity
B0019082biological_processviral protein processing
C0008233molecular_functionpeptidase activity
C0019082biological_processviral protein processing
D0008233molecular_functionpeptidase activity
D0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE K36 A 401
ChainResidue
AHIS41
AGLU165
AHIS171
AGLN187
AHOH513
APHE139
AILE140
AGLY142
ATHR143
ACYS144
AHIS162
AHIS163
ALEU164

site_idAC2
Number of Residues14
DetailsBINDING SITE FOR RESIDUE K36 B 401
ChainResidue
BHIS41
BPHE139
BILE140
BGLY142
BTHR143
BCYS144
BHIS162
BHIS163
BLEU164
BGLU165
BHIS171
BGLN187
BPRO188
BHOH548

site_idAC3
Number of Residues14
DetailsBINDING SITE FOR RESIDUE K36 C 401
ChainResidue
CTHR47
CILE51
CPHE139
CILE140
CGLY142
CTHR143
CCYS144
CHIS162
CHIS163
CLEU164
CGLU165
CHIS171
CGLN187
CHOH523

site_idAC4
Number of Residues12
DetailsBINDING SITE FOR RESIDUE K36 D 401
ChainResidue
DPHE139
DILE140
DALA141
DTHR143
DCYS144
DHIS162
DHIS163
DLEU164
DGLU165
DHIS171
DGLN187
DPRO188

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PG4 D 402
ChainResidue
AARG19
ASER21
DARG267
DLYS270
DHOH502
DHOH519

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsActive site: {"description":"For 3CL-PRO activity","evidences":[{"source":"PROSITE-ProRule","id":"PRU00772","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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