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4ERF

crystal structure of MDM2 (17-111) in complex with compound 29 (AM-8553)

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0043066biological_processnegative regulation of apoptotic process
A0051726biological_processregulation of cell cycle
C0005634cellular_componentnucleus
C0043066biological_processnegative regulation of apoptotic process
C0051726biological_processregulation of cell cycle
E0005634cellular_componentnucleus
E0043066biological_processnegative regulation of apoptotic process
E0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 0R3 A 201
ChainResidue
ALEU54
AHOH335
AILE61
ATYR67
AVAL93
ALYS94
AHIS96
AILE99
ATYR100
AHOH325

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE 0R3 C 201
ChainResidue
AARG97
CLEU54
CGLY58
CVAL93
CLYS94
CHIS96
CILE99
CHOH323

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE 0R3 E 201
ChainResidue
ELEU54
EILE61
EVAL93
ELYS94
EHIS96
ETYR100

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues249
DetailsDomain: {"description":"SWIB/MDM2","evidences":[{"source":"PROSITE-ProRule","id":"PRU01273","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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