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4CFL

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH LY303511

Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 8DQ A 1169
ChainResidue
ATRP81
AHOH2239
AHOH2287
APRO82
AVAL87
ALEU92
ALEU94
AASN140
AILE146
AGOL1171
AHOH2173

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1170
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1171
ChainResidue
ALYS57
AASP144
AASP145
AILE146
A8DQ1169
AHOH2288

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

225158

PDB entries from 2024-09-18

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