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4BVV

Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV.

Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE CPF A 1081
ChainResidue
APHE3
ALEU71
APHE72
ASER34
ATHR35
AASP55
AASP57
AILE58
AASN59
ATRP62
ATYR64

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1082
ChainResidue
AASP0
ATYR9
ALYS12
ALYS13

Functional Information from PROSITE/UniProt
site_idPS00021
Number of Residues14
DetailsKRINGLE_1 Kringle domain signature. YCRNpdgdingpWC
ChainResidueDetails
ATYR50-CYS63

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues80
DetailsDomain: {"description":"Kringle 16","evidences":[{"source":"PROSITE-ProRule","id":"PRU00121","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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