4BV5
Identification of small molecule inhibitors selective for apo(a) kringles KIV-7, KIV-10 and KV.
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 12 |
Details | BINDING SITE FOR RESIDUE 5C3 A 1081 |
Chain | Residue |
A | HIS33 |
B | ASP67 |
B | PRO68 |
B | SER69 |
A | GLN34 |
A | ARG35 |
A | ASP55 |
A | ASP57 |
A | TRP62 |
A | PHE64 |
A | ARG71 |
A | TRP72 |
site_id | AC2 |
Number of Residues | 11 |
Details | BINDING SITE FOR RESIDUE 5C3 B 1081 |
Chain | Residue |
A | ASP67 |
A | PRO68 |
A | SER69 |
B | HIS33 |
B | GLN34 |
B | ARG35 |
B | ASP55 |
B | ASP57 |
B | TRP62 |
B | ARG71 |
B | TRP72 |
Functional Information from PROSITE/UniProt
site_id | PS00021 |
Number of Residues | 13 |
Details | KRINGLE_1 Kringle domain signature. YCRNpdadtgp.WC |
Chain | Residue | Details |
A | TYR50-CYS63 |