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4AZI

Differential inhibition of the tandem GH20 catalytic modules in the pneumococcal exo-beta-D-N-acetylglucosaminidase, StrH

Functional Information from GO Data
ChainGOidnamespacecontents
A0004553molecular_functionhydrolase activity, hydrolyzing O-glycosyl compounds
A0005975biological_processcarbohydrate metabolic process
B0004553molecular_functionhydrolase activity, hydrolyzing O-glycosyl compounds
B0005975biological_processcarbohydrate metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE OAN A 2038
ChainResidue
AARG641
AASP953
AEDO2041
AHOH3047
AHOH3565
AHOH3566
AHIS742
AASP804
AGLU805
ATRP872
ATYR902
AILE904
ATYR914
ATRP951

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2039
ChainResidue
AHIS625
AASN1020
AASN1022
ALYS1023
AHOH3520

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2040
ChainResidue
AGLN716
ALYS795
AHOH3113
AHOH3199
AHOH3569

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 2041
ChainResidue
AHIS742
AGLU805
AASN808
AOAN2038
AHOH3016
AHOH3565

site_idAC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE BR A 2042
ChainResidue
APHE915
ALEU916
ALYS917

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE BR A 2043
ChainResidue
APRO955
ASER956

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE BR A 2044
ChainResidue
AGLN823
ATYR825
AGLY826

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE BCN A 2045
ChainResidue
ATHR834
AALA837
AMET838
AGLU841
AHOH3230

site_idAC9
Number of Residues15
DetailsBINDING SITE FOR RESIDUE OAN B 2040
ChainResidue
BARG641
BHIS742
BASP804
BGLU805
BPHE849
BTRP872
BTYR902
BILE904
BTRP913
BTYR914
BTRP951
BASP953
BEDO2043
BBCN2046
BHOH3049

site_idBC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO B 2041
ChainResidue
BARG954
BPRO955
BHOH3445

site_idBC2
Number of Residues1
DetailsBINDING SITE FOR RESIDUE EDO B 2042
ChainResidue
BHOH3131

site_idBC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO B 2043
ChainResidue
BARG641
BHIS742
BGLU805
BASN808
BOAN2040
BBCN2046

site_idBC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE BR B 2044
ChainResidue
BTYR854
BGLN862
BLYS890
BHOH3325

site_idBC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE BCN B 2045
ChainResidue
BHIS974
BHOH3385
BHOH3476

site_idBC6
Number of Residues8
DetailsBINDING SITE FOR RESIDUE BCN B 2046
ChainResidue
BALA813
BTRP913
BTYR914
BOAN2040
BEDO2043
BHOH3187
BHOH3534
BHOH3535

221051

PDB entries from 2024-06-12

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