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4AZG

Differential inhibition of the tandem GH20 catalytic modules in the pneumococcal exo-beta-D-N-acetylglucosaminidase, StrH

Functional Information from GO Data
ChainGOidnamespacecontents
A0004553molecular_functionhydrolase activity, hydrolyzing O-glycosyl compounds
A0005975biological_processcarbohydrate metabolic process
B0004553molecular_functionhydrolase activity, hydrolyzing O-glycosyl compounds
B0005975biological_processcarbohydrate metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE OAN B 2041
ChainResidue
BARG641
BTRP951
BASP953
BHOH3040
BHIS742
BASP804
BGLU805
BTRP872
BTRP876
BTYR879
BTYR902
BILE904

site_idAC2
Number of Residues13
DetailsBINDING SITE FOR RESIDUE OAN A 2040
ChainResidue
AARG641
AHIS742
AASP804
AGLU805
ATRP872
ATRP876
ATYR879
ATYR902
AILE904
ATRP951
AASP953
AACT2043
AHOH3044

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ACT B 2042
ChainResidue
BTYR854
BGLN862
BLYS865
BLYS890

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ACT B 2043
ChainResidue
BTYR705
BASP744
BHOH3062
BHOH3065

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE ACT A 2041
ChainResidue
AGLN1039
AHOH3271

site_idAC6
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ACT A 2042
ChainResidue
ATYR854
AGLN862
ALYS865
ALYS890
AHOH3176

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ACT A 2043
ChainResidue
AARG641
AGLU805
AASN808
AOAN2040

site_idAC8
Number of Residues3
DetailsBINDING SITE FOR RESIDUE ACT B 2044
ChainResidue
BARG641
BGLU805
BASN808

site_idAC9
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2044
ChainResidue
AGLN648
ATYR959
AGLU961

site_idBC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE EDO B 2045
ChainResidue
BSER657
BGLY660
BTYR661
BLYS729
BASP730
BILE731
BARG980
BHOH3030
BHOH3031
BHOH3273

site_idBC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 2046
ChainResidue
BILE904
BLEU905
BGLY906
BGLN907
BARG954

site_idBC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 2045
ChainResidue
ATYR705
AASP744
AHOH3067

site_idBC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO B 2047
ChainResidue
BHIS761
BASP771
BLEU772
BTYR806

site_idBC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2046
ChainResidue
AALA760
AHIS761
AASP771
ALEU772
ATYR806

site_idBC6
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2047
ChainResidue
AGLU751
AGLY754
ALYS756
AASN757
AHOH3273

site_idBC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 2048
ChainResidue
ATYR903
AGLN907
ALEU916
AGLU963
AHOH3185

site_idBC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 2048
ChainResidue
BGLY906
BARG954
BALA957
BGLU958
BHOH3227

224931

PDB entries from 2024-09-11

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