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4ALG

N-Terminal Bromodomain of Human BRD2 With IBET-151

Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ACT A 1144
ChainResidue
AARG54
ALYS69
AHOH2024
AHOH2053

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE GOL A 1145
ChainResidue
AHOH2102
AHOH2125
AHOH2126
AASP58
AHIS68
AASP114
AASP115
AHOH2042

site_idAC3
Number of Residues12
DetailsBINDING SITE FOR RESIDUE 1GH A 1146
ChainResidue
ATRP51
APRO52
APHE53
ALEU62
ALEU64
AHIS68
ALYS72
AASN110
AILE116
AHOH2034
AHOH2055
AHOH2126

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA50-TYR109

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
ChainResidueDetails
AASP66
ATYR109
AASN110
ALYS111

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000269|PubMed:20048151, ECO:0007744|PDB:2DVQ, ECO:0007744|PDB:2DVS
ChainResidueDetails
AASP114
AASP115

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PDB entries from 2025-06-18

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