Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

4A9N

N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH N-cyclopropyl-5-(3,5- dimethyl-1,2-oxazol-4-yl)-2-methylbenzene-1-sulfonamide

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1187
ChainResidue
AHIS114
ALYS118
AHOH2054
BGLN119
BARG129
BASP144
BHOH2052

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1188
ChainResidue
ALYS118
AGLN119
AASN151
AILE116
AILE117

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1189
ChainResidue
AGLN143
AHOH2082
BLYS118

site_idAC4
Number of Residues10
DetailsBINDING SITE FOR RESIDUE A9N A 1190
ChainResidue
ATRP97
APRO98
APHE99
ALEU108
ALEU110
AASN156
AHOH2051
AHOH2094
AHOH2121
BGLN94

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1191
ChainResidue
AARG100
AHOH2011
AHOH2013
AHOH2015

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1192
ChainResidue
ATHR125
AARG128
AARG129

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 1187
ChainResidue
AGLN94
ATRP97
AMET165
BGLN94
BTRP97

site_idAC8
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO B 1188
ChainResidue
ALYS171
BGLN143
BASN146

site_idAC9
Number of Residues9
DetailsBINDING SITE FOR RESIDUE A9N B 1189
ChainResidue
AGLN94
BTRP97
BPRO98
BPHE99
BLEU108
BASN156
BHOH2028
BHOH2076
BHOH2088

site_idBC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 B 1190
ChainResidue
BTHR125
BARG128
BARG129

site_idBC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE DMS C 1183
ChainResidue
CASN156
CHOH2026

site_idBC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO C 1184
ChainResidue
CARG129
CASP144
CHOH2039

site_idBC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 C 1185
ChainResidue
BARG100
CARG128
CASN132
CTYR134
CHOH2037
CHOH2067
CHOH2068

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA96-TYR155

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsBINDING: BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
ChainResidueDetails
AASP112
CTYR155
CASN156
CLYS157
ATYR155
AASN156
ALYS157
BASP112
BTYR155
BASN156
BLYS157
CASP112

site_idSWS_FT_FI2
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:20048151, ECO:0007744|PDB:2DVQ, ECO:0007744|PDB:2DVS
ChainResidueDetails
AASP160
AASP161
BASP160
BASP161
CASP160
CASP161

222624

PDB entries from 2024-07-17

PDB statisticsPDBj update infoContact PDBjnumon