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4A9L

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH 1,3-DIMETHYL-6-(MORPHOLINE- 4-SULFONYL)-1,2,3,4-TETRAHYDROQUINAZOLIN-2-ONE

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1168
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH2235

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1169
ChainResidue
AHOH2117
AHOH2126
ATRP81
AGLN85
AASP96

site_idAC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 1170
ChainResidue
ALEU67
AGLU115

site_idAC4
Number of Residues11
DetailsBINDING SITE FOR RESIDUE P9L A 1171
ChainResidue
ATRP81
APRO82
APHE83
ALEU94
ALYS99
ATYR139
AASN140
AILE146
AMET149
AHOH2130
AHOH2237

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE NO3 A 1172
ChainResidue
ALYS57
AASN116
AASN117
AASP145
AHOH2160

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE NO3 A 1173
ChainResidue
ATHR60
AGLN62
AASN121
AALA122
AGLU167
AHOH2165

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

222415

PDB entries from 2024-07-10

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