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4A2J

PR X-Ray structures in agonist conformations reveal two different mechanisms for partial agonism in 11beta-substituted steroids

Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE AS0 A 1000
ChainResidue
ALEU715
AARG766
APHE778
APHE794
ALEU797
AMET801
ACYS891
AMET909
ALEU718
AASN719
AGLY722
AGLU723
AGLN725
ALEU726
ATRP755
AMET759

site_idAC2
Number of Residues16
DetailsBINDING SITE FOR RESIDUE AS0 B 1000
ChainResidue
BLEU715
BLEU718
BASN719
BLEU721
BGLY722
BGLU723
BGLN725
BLEU726
BTRP755
BMET759
BARG766
BPHE778
BMET801
BTYR890
BCYS891
BMET909

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1934
ChainResidue
APRO737
AGLY738
AARG740
AASN741
AHOH2010

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9620806","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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