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3WPN

Kinesin spindle protein Eg5 in complex with ATP-competitive inhibitor PVZB1194

Functional Information from GO Data
ChainGOidnamespacecontents
A0003777molecular_functionmicrotubule motor activity
A0005524molecular_functionATP binding
A0007018biological_processmicrotubule-based movement
A0008017molecular_functionmicrotubule binding
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE B4S A 401
ChainResidue
ATYR104
ALEU369
AGLU253
ALEU292
ALEU293
ALEU295
AILE332
AALA334
ATYR352
AALA353

Functional Information from PROSITE/UniProt
site_idPS00411
Number of Residues12
DetailsKINESIN_MOTOR_1 Kinesin motor domain signature. GKLnLVDLAGSE
ChainResidueDetails
AGLY259-GLU270

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00283
ChainResidueDetails
AGLY105

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0007744|PubMed:19608861
ChainResidueDetails
ALYS146

237735

PDB entries from 2025-06-18

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