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3WNG

Cyclic hexapeptide PKIDNp in complex with HIV-1 integrase

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD A 1001
ChainResidue
ACYS65
AHIS67
AGLU92
BASP131

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD A 1002
ChainResidue
BHOH408
ACYS65
AGLU92
AASP116
ACL1003
AHOH1101

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 1003
ChainResidue
ACYS65
AASP116
AASN120
ACD1002

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1004
ChainResidue
ALYS71
AARG166
AGLU170
AHIS171
ALEU172
AHOH1117
AHOH1127

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1005
ChainResidue
ATHR66
AHIS67
AGLU152
ALYS159
BARG127

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1006
ChainResidue
AGLY123
AALA124
ATHR125
AHOH1107
AHOH1108
AHOH1119
AHOH1125

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD B 301
ChainResidue
AASP131
BCYS65
BHIS67
BGLU92

site_idAC8
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CD B 302
ChainResidue
AHOH1105
BCYS65
BGLU92
BASP116
BCL303
BHOH401

site_idAC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL B 303
ChainResidue
BCYS65
BASP116
BASN120
BCD302

site_idBC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 304
ChainResidue
BLYS71
BARG166
BGLU170
BHIS171
BLEU172
BHOH418
BHOH435

site_idBC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 305
ChainResidue
BGLY123
BALA124
BTHR125
BHOH407
BHOH419
BHOH428

site_idBC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 306
ChainResidue
BTHR66
BHIS67
BGLU152
BLYS159

site_idBC4
Number of Residues8
DetailsBINDING SITE FOR CHAIN C OF PKIDN(DPR) PEPTIDE
ChainResidue
AGLN95
ATHR125
BASP167
BGLN168
BALA169
BGLU170
BHIS171
BTHR174

site_idBC5
Number of Residues9
DetailsBINDING SITE FOR CHAIN D OF PKIDN(DPR) PEPTIDE
ChainResidue
AASP167
AGLN168
AALA169
AGLU170
AHIS171
ATHR174
BGLN95
BTHR125
DHOH101

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING:
ChainResidueDetails
AASP64
AASP116
BASP64
BASP116

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152
BGLU152

224004

PDB entries from 2024-08-21

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