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3WMH

Human PPAR gamma ligand binding domain in complex with a gammma selective synthetic partial agonist MEKT75

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues17
DetailsBINDING SITE FOR RESIDUE JJA A 901
ChainResidue
APHE264
AILE326
ATYR327
ALEU330
AMET348
APHE363
ALYS367
AHIS449
AHOH1037
AHIS266
AARG280
AILE281
APHE282
AGLY284
ACYS285
AARG288
ASER289

site_idAC2
Number of Residues12
DetailsBINDING SITE FOR RESIDUE JJA B 901
ChainResidue
BHIS266
BARG280
BILE281
BPHE282
BCYS285
BARG288
BSER289
BILE326
BTYR327
BPHE363
BMET364
BHIS449

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
ChainResidueDetails
AGLN286
AHIS323
AHIS449
ATYR473
BGLN286
BHIS323
BHIS449
BTYR473

site_idSWS_FT_FI2
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224
BLYS224

219140

PDB entries from 2024-05-01

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