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3UH4

TANKYRASE-1 complexed with NVP-XAV939

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2001
ChainResidue
ACYS1234
AHIS1237
ACYS1242
ACYS1245

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE XAV A 1
ChainResidue
ATYR1213
APHE1214
ASER1221
ATYR1224
AASN1285
AHIS1184
AGLY1185
ASER1186
APRO1187
APHE1188

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1328
ChainResidue
AHOH162
AHIS1176
AHIS1177
AASN1178
BHIS1176

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 3
ChainResidue
AHOH79
AARG1130
AHIS1132
AARG1133
ALYS1220

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 5
ChainResidue
AHOH12
AASN1143
APRO1313
AGLU1314

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 A 6
ChainResidue
AARG1149
AHIS1246

site_idAC7
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 11
ChainResidue
AHOH229
AHIS1184
ASER1186
AILE1192
APHE1197
AASP1198
AHIS1201

site_idAC8
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 2001
ChainResidue
BCYS1234
BHIS1237
BCYS1242
BCYS1245

site_idAC9
Number of Residues13
DetailsBINDING SITE FOR RESIDUE XAV B 1
ChainResidue
BHOH310
BHIS1184
BGLY1185
BSER1186
BPRO1187
BHIS1201
BTYR1203
BTYR1213
BPHE1214
BSER1221
BTYR1224
BILE1228
BGLU1291

site_idBC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 2
ChainResidue
BHOH113
BARG1130
BHIS1132
BARG1133
BLYS1220

site_idBC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 B 7
ChainResidue
BHIS1176
BHIS1177
BASN1178

site_idBC3
Number of Residues1
DetailsBINDING SITE FOR RESIDUE SO4 B 8
ChainResidue
BARG1253

site_idBC4
Number of Residues11
DetailsBINDING SITE FOR RESIDUE GOL B 9
ChainResidue
BHOH86
BHOH153
BHIS1184
BSER1186
BILE1192
BASP1198
BHIS1201
BALA1202
BTYR1203
BGLY1211
BILE1212

site_idBC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL B 10
ChainResidue
BHOH236
BHOH310
BILE1204

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PDB entries from 2024-10-16

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