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3U78

E67-2 selectively inhibits KIAA1718, a human histone H3 lysine 9 Jumonji demethylase

Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE AKG A 701
ChainResidue
AASN224
ANI702
AE67707
AHOH801
AHOH843
AILE226
ATHR279
AHIS282
AASP284
ATYR292
ALYS299
AHIS354
AVAL356

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE NI A 702
ChainResidue
AHIS282
AASP284
AHIS354
AAKG701
AHOH801

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE CL A 703
ChainResidue
ASER249
ATRP250
AVAL251
APHE369
ALEU370

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 704
ChainResidue
AGLU309
AARG313
AASP333

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 705
ChainResidue
ALYS153
AHOH873

site_idAC6
Number of Residues1
DetailsBINDING SITE FOR RESIDUE EDO A 706
ChainResidue
AASP167

site_idAC7
Number of Residues9
DetailsBINDING SITE FOR RESIDUE E67 A 707
ChainResidue
AGLN200
AASP202
ALYS204
AASP280
AASP284
APHE285
APRO391
AASP392
AAKG701

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
ATHR279
ALYS299

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00538, ECO:0000269|PubMed:20023638
ChainResidueDetails
AHIS282
AASP284
AHIS354

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PDB entries from 2024-07-17

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