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3TU1

Exhaustive Fluorine Scanning towards Potent p53-MDM2 Antagonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0043066biological_processnegative regulation of apoptotic process
A0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE 07G A 1
ChainResidue
AHOH3
ATYR100
AHOH138
AHOH165
ALEU54
AGLY58
AILE61
AMET62
ATYR67
AVAL93
AHIS96
AILE99

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues83
DetailsDomain: {"description":"SWIB/MDM2","evidences":[{"source":"PROSITE-ProRule","id":"PRU01273","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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