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3SMJ

Human poly(ADP-ribose) polymerase 14 (Parp14/Artd8) - catalytic domain in complex with a pyrimidine-like inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE FDR A 1
ChainResidue
AHOH289
AGLN1683
AHIS1601
AGLY1602
ATYR1633
AALA1635
ATYR1640
ASER1641
ATYR1646
APRO1682

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1721
ChainResidue
AHOH2
AHOH65
AHOH264
AHIS1601
ATHR1603
AARG1618

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE FDR B 2
ChainResidue
BHOH88
BHIS1601
BGLY1602
BGLY1622
BTYR1633
BSER1641
BTYR1646

222415

PDB entries from 2024-07-10

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