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3SFX

Cryptococcus neoformans protein farnesyltransferase in complex with FPT-II and tipifarnib

Functional Information from GO Data
ChainGOidnamespacecontents
A0008318molecular_functionprotein prenyltransferase activity
A0018342biological_processprotein prenylation
B0003824molecular_functioncatalytic activity
B0005965cellular_componentprotein farnesyltransferase complex
B0008318molecular_functionprotein prenyltransferase activity
B0018343biological_processprotein farnesylation
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 521
ChainResidue
BASP323
BCYS325
BHIS410
BJAN526

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 3FX B 522
ChainResidue
BARG493
BASN495
BHOH1774
BHOH1900
BHOH2460
BTYR58
BASP100
BGLY489
BLYS490
BASP491

site_idAC3
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 3FX B 523
ChainResidue
BARG62
BLYS63
BGLN64
BGLU65
BPHE74
BPHE75
BHOH1877
BHOH1972
BHOH1994
BHOH2102

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE 3FX B 524
ChainResidue
BSER123
BPRO124
BLYS125
BALA133
BASN134
BSER135
BGLN136

site_idAC5
Number of Residues17
DetailsBINDING SITE FOR RESIDUE FII B 525
ChainResidue
AHOH2096
BTRP90
BLEU141
BARG197
BHIS266
BGLY268
BTYR269
BCYS272
BARG317
BLYS320
BTYR326
BTRP329
BJAN526
BHOH2087
BHOH2092
BHOH2101
BHOH2547

site_idAC6
Number of Residues14
DetailsBINDING SITE FOR RESIDUE JAN B 526
ChainResidue
BLEU84
BTRP94
BARG197
BASP323
BCYS325
BTYR326
BASP407
BTYR409
BHIS410
BZN521
BFII525
BHOH2588
BHOH2773
BHOH2869

site_idAC7
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 B 527
ChainResidue
ATYR74
BALA86
BSER87
BTRP90
BHIS139
BLEU141
BPRO142
BHOH2111

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PDB entries from 2024-07-31

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