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3DR1

Side-chain fluorine atoms of non-steroidal vitamin D3 analogs stabilize helix 12 of vitamin D receptor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE C5D A 500
ChainResidue
ATYR175
AHIS333
ALEU341
AHIS423
ATYR427
ALEU430
ALEU440
APHE448
ATYR179
ALEU255
ASER265
AARG302
ASER303
ASER306
ACYS316
AALA331

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
AHIS333
AHIS423
ALEU255
AILE299

218500

PDB entries from 2024-04-17

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