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3BQD

Doubling the Size of the Glucocorticoid Receptor Ligand Binding Pocket by Deacylcortivazol

Functional Information from PDB Data
site_idAC1
Number of Residues18
DetailsBINDING SITE FOR RESIDUE DAY A 301
ChainResidue
ALEU563
ALEU608
AARG611
APHE623
AGLN642
ALEU732
ATYR735
ACYS736
ATHR739
AILE747
AASN564
ALEU566
AGLY567
AGLN570
AMET601
AMET604
AALA605
AALA607

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
ChainResidueDetails
ALYS703

225946

PDB entries from 2024-10-09

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