3AVR
Catalytic fragment of UTX/KDM6A bound with histone H3K27me3 peptide, N-oxyalylglycine, and Ni(II)
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 12 |
Details | BINDING SITE FOR RESIDUE OGA A 1501 |
Chain | Residue |
A | HOH63 |
A | ALA1238 |
A | NI1503 |
B | M3L27 |
A | LYS1137 |
A | THR1143 |
A | HIS1146 |
A | GLU1148 |
A | SER1154 |
A | ASN1156 |
A | TRP1166 |
A | HIS1226 |
site_id | AC2 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE ZN A 1502 |
Chain | Residue |
A | CYS1331 |
A | CYS1334 |
A | CYS1358 |
A | CYS1361 |
site_id | AC3 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE NI A 1503 |
Chain | Residue |
A | HOH265 |
A | HIS1146 |
A | GLU1148 |
A | HIS1226 |
A | OGA1501 |
site_id | AC4 |
Number of Residues | 2 |
Details | BINDING SITE FOR RESIDUE EDO A 1 |
Chain | Residue |
A | HOH295 |
A | SER1120 |
site_id | AC5 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE EDO A 2 |
Chain | Residue |
A | HOH115 |
A | HOH198 |
A | GLU946 |
A | MET1291 |
site_id | AC6 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE EDO A 3 |
Chain | Residue |
A | HOH343 |
A | PRO932 |
A | LYS933 |
A | ASN1204 |
site_id | AC7 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO A 4 |
Chain | Residue |
A | HOH60 |
A | HOH99 |
A | HOH104 |
A | ILE889 |
A | TYR890 |
A | PRO891 |
A | THR940 |
site_id | AC8 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO A 5 |
Chain | Residue |
A | HOH55 |
A | HOH210 |
A | GLN1039 |
A | ALA1040 |
A | TRP1233 |
site_id | AC9 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE EDO A 6 |
Chain | Residue |
A | HOH275 |
A | HOH296 |
A | THR1030 |
A | LYS1034 |
A | TYR1035 |
A | LYS1083 |
site_id | BC1 |
Number of Residues | 2 |
Details | BINDING SITE FOR RESIDUE EDO A 7 |
Chain | Residue |
A | ALA1108 |
A | ARG1111 |
site_id | BC2 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE EDO A 8 |
Chain | Residue |
A | HOH329 |
A | THR961 |
A | ASN1221 |
A | ALA1222 |
A | THR1245 |
A | CYS1247 |
site_id | BC3 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO A 9 |
Chain | Residue |
A | HOH56 |
A | HOH368 |
A | LEU981 |
A | GLY982 |
A | ILE1159 |
site_id | BC4 |
Number of Residues | 1 |
Details | BINDING SITE FOR RESIDUE CL A 1402 |
Chain | Residue |
A | ARG1322 |
site_id | BC5 |
Number of Residues | 2 |
Details | BINDING SITE FOR RESIDUE CL A 1403 |
Chain | Residue |
A | SER1114 |
A | ALA1115 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 1 |
Details | MOD_RES: Citrulline; alternate => ECO:0000269|PubMed:15345777, ECO:0000269|PubMed:16497732, ECO:0000269|PubMed:16567635 |
Chain | Residue | Details |
B | ARG17 | |
A | GLU1148 | |
A | HIS1226 | |
A | CYS1331 | |
A | CYS1334 | |
A | CYS1358 | |
A | CYS1361 |
site_id | SWS_FT_FI2 |
Number of Residues | 1 |
Details | MOD_RES: N6-methyllysine; alternate => ECO:0000269|PubMed:16267050, ECO:0000269|PubMed:17194708 |
Chain | Residue | Details |
B | LYS18 |
site_id | SWS_FT_FI3 |
Number of Residues | 1 |
Details | MOD_RES: N6-methyllysine; alternate => ECO:0000269|PubMed:17194708 |
Chain | Residue | Details |
B | LYS23 |
site_id | SWS_FT_FI4 |
Number of Residues | 1 |
Details | MOD_RES: Citrulline => ECO:0000269|PubMed:16567635 |
Chain | Residue | Details |
B | ARG26 |
site_id | SWS_FT_FI5 |
Number of Residues | 1 |
Details | MOD_RES: N6-methyllysine; alternate => ECO:0000269|PubMed:16185088, ECO:0000269|PubMed:16267050, ECO:0000269|PubMed:16627869, ECO:0000269|PubMed:17194708 |
Chain | Residue | Details |
B | M3L27 |
site_id | SWS_FT_FI6 |
Number of Residues | 1 |
Details | MOD_RES: Phosphoserine; alternate; by AURKB, AURKC and RPS6KA5 => ECO:0000269|PubMed:10464286, ECO:0000269|PubMed:11856369, ECO:0000269|PubMed:15681610, ECO:0000269|PubMed:15684425, ECO:0000269|PubMed:16185088, ECO:0000269|PubMed:16457588 |
Chain | Residue | Details |
B | SER28 |
site_id | SWS_FT_FI7 |
Number of Residues | 1 |
Details | MOD_RES: N6-methyllysine; alternate => ECO:0000269|PubMed:15983376, ECO:0000269|PubMed:16185088, ECO:0000269|PubMed:16267050, ECO:0000269|PubMed:16627869, ECO:0000269|PubMed:17194708 |
Chain | Residue | Details |
B | LYS36 |
site_id | SWS_FT_FI8 |
Number of Residues | 1 |
Details | MOD_RES: N6-methyllysine => ECO:0000269|PubMed:15983376 |
Chain | Residue | Details |
B | LYS37 |
site_id | SWS_FT_FI9 |
Number of Residues | 1 |
Details | LIPID: N6-decanoyllysine => ECO:0000269|PubMed:35939806 |
Chain | Residue | Details |
B | LYS18 |