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2ZNO

Human PPAR gamma ligand binding domain in complex with a synthetic agonist TIPP703

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE S44 A 901
ChainResidue
ALEU255
AMET348
AMET364
AHIS449
ATYR473
AARG280
AILE281
APHE282
ACYS285
AARG288
ASER289
AHIS323
AILE341

site_idAC2
Number of Residues14
DetailsBINDING SITE FOR RESIDUE S44 B 902
ChainResidue
BLEU255
BARG280
BPHE282
BCYS285
BGLN286
BARG288
BSER289
BHIS323
BTYR327
BLEU330
BILE341
BPHE363
BMET364
BHIS449

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
ChainResidueDetails
AGLN286
AHIS323
AHIS449
ATYR473
BGLN286
BHIS323
BHIS449
BTYR473

site_idSWS_FT_FI2
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224
BLYS224

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PDB entries from 2024-07-24

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