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2IW5

Structural Basis for CoREST-Dependent Demethylation of Nucleosomes by the Human LSD1 Histone Demethylase

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0016491molecular_functionoxidoreductase activity
A0050660molecular_functionflavin adenine dinucleotide binding
Functional Information from PDB Data
site_idAC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A1838
ChainResidue
AASP754
ACL1843

site_idAC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A1843
ChainResidue
AARG750
ACL1838

site_idAC3
Number of Residues37
DetailsBINDING SITE FOR RESIDUE FAD A 900
ChainResidue
AGLU308
AALA309
AARG310
AGLY314
AGLY315
AARG316
AVAL317
ALEU329
AGLY330
AALA331
AMET332
AVAL333
ATHR588
AALA589
AVAL590
ATHR624
ALEU625
APRO626
ATRP751
ATRP756
ASER760
ATYR761
AGLY800
AGLU801
AALA809
ATHR810
AVAL811
AALA814
AHOH2034
AHOH2042
AHOH2075
AHOH2076
AGLY285
AGLY287
AVAL288
ASER289
ALEU307

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A1839
ChainResidue
AARG526
ALEU544
AARG688

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE GOL A1840
ChainResidue
AGLN358
AASN535

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:21406692, ECO:0007744|PubMed:23186163
ChainResidueDetails
BASN460
AGLU308
AARG310
AARG316
AMET332
AGLU801
ATHR810

site_idSWS_FT_FI2
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
BLYS297
BGLU466

site_idSWS_FT_FI3
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS442
ALYS469

site_idSWS_FT_FI4
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000305|PubMed:25018020
ChainResidueDetails
ALYS503

218853

PDB entries from 2024-04-24

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