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2FSZ

A second binding site for hydroxytamoxifen within the coactivator-binding groove of estrogen receptor beta

Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE OHT A 101
ChainResidue
AMET295
AGLY472
ALEU476
BHOH27
BPRO486
ALEU298
ATHR299
AASP303
AGLU305
AMET336
AARG346
AILE373
ALEU380

site_idAC2
Number of Residues14
DetailsBINDING SITE FOR RESIDUE OHT B 102
ChainResidue
APRO486
BMET295
BLEU298
BALA302
BASP303
BGLU305
BLEU306
BMET336
BMET340
BARG346
BILE373
BLEU380
BGLY472
BLEU476

site_idAC3
Number of Residues13
DetailsBINDING SITE FOR RESIDUE OHT A 103
ChainResidue
ALEU306
AILE310
ALYS314
AGLN327
AVAL328
ALEU331
AGLU332
ATRP335
BOHT104
BLEU490
BMET494
BVAL499
BARG501

site_idAC4
Number of Residues13
DetailsBINDING SITE FOR RESIDUE OHT B 104
ChainResidue
AOHT103
ALEU490
AMET494
AARG501
BHOH32
BLEU306
BILE310
BLEU324
BGLN327
BVAL328
BLEU331
BGLU332
BTRP335

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PDB entries from 2024-07-24

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