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2AIX

X-ray structure of the GLUR2 ligand-binding core (S1S2J) in complex with (s)-thio-atpa at 2.2 a resolution.

Functional Information from GO Data
ChainGOidnamespacecontents
A0015276molecular_functionligand-gated monoatomic ion channel activity
A0016020cellular_componentmembrane
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE U1K A 261
ChainResidue
AGLU10
ATHR171
AGLU190
AMET193
AHOH269
AHOH276
ATYR58
APRO86
ALEU87
ATHR88
AARG93
AGLY138
ASER139
ATHR140

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues40
DetailsTRANSMEM: Helical
ChainResidueDetails
AALA131-VAL151
AASP204-GLY224

site_idSWS_FT_FI2
Number of Residues31
DetailsTOPO_DOM: Cytoplasmic
ChainResidueDetails
APHE152-VAL178
AGLU198-CYS203

site_idSWS_FT_FI3
Number of Residues15
DetailsINTRAMEM: Helical; Pore-forming
ChainResidueDetails
AARG179-ASN194

site_idSWS_FT_FI4
Number of Residues2
DetailsINTRAMEM:
ChainResidueDetails
AGLU195-ILE197

site_idSWS_FT_FI5
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:11086992, ECO:0000269|PubMed:16483599, ECO:0007744|PDB:1FTJ, ECO:0007744|PDB:2CMO
ChainResidueDetails
APRO86
ATHR88
AARG93
ASER139
ATHR140
AGLU190

site_idSWS_FT_FI6
Number of Residues3
DetailsSITE: Interaction with the cone snail toxin Con-ikot-ikot => ECO:0000269|PubMed:25103405
ChainResidueDetails
AARG61
AARG145
ALYS237

site_idSWS_FT_FI7
Number of Residues1
DetailsSITE: Crucial to convey clamshell closure to channel opening => ECO:0000269|PubMed:25103405
ChainResidueDetails
AILE118

site_idSWS_FT_FI8
Number of Residues1
DetailsMOD_RES: Phosphoserine; by PKC => ECO:0000269|PubMed:8848293
ChainResidueDetails
ASER147

site_idSWS_FT_FI9
Number of Residues1
DetailsMOD_RES: Phosphoserine; by PKG => ECO:0000269|PubMed:8848293
ChainResidueDetails
ASER181

site_idSWS_FT_FI10
Number of Residues1
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
AILE197

site_idSWS_FT_FI11
Number of Residues1
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
AASN0

222036

PDB entries from 2024-07-03

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