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1S9Q

crystal structure of the ligand-binding domain of the estrogen-related receptor gamma in complex with 4-hydroxytamoxifen

Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE OHT A 200
ChainResidue
ALEU268
AALA431
AHIS434
APHE435
AILE438
ACHD459
ACYS269
AALA272
AASP273
AGLU275
ATRP305
ALEU309
AARG316
ATYR326

site_idAC2
Number of Residues14
DetailsBINDING SITE FOR RESIDUE OHT B 459
ChainResidue
BLEU268
BCYS269
BALA272
BASP273
BGLU275
BTRP305
BLEU309
BVAL313
BARG316
BTYR326
BALA431
BHIS434
BPHE435
BCHD500

site_idAC3
Number of Residues8
DetailsBINDING SITE FOR RESIDUE CHD A 459
ChainResidue
AOHT200
AASP273
ALEU276
AVAL277
AILE280
ATRP305
AHIS447
APHE450

site_idAC4
Number of Residues9
DetailsBINDING SITE FOR RESIDUE CHD B 500
ChainResidue
BASP273
BLEU276
BILE280
BTRP305
BPRO445
BMET446
BLEU449
BPHE450
BOHT459

224201

PDB entries from 2024-08-28

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