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1PQ6

HUMAN LXR BETA HORMONE RECEPTOR / GW3965 COMPLEX

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006629biological_processlipid metabolic process
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006629biological_processlipid metabolic process
C0003677molecular_functionDNA binding
C0004879molecular_functionnuclear receptor activity
C0006629biological_processlipid metabolic process
D0003677molecular_functionDNA binding
D0004879molecular_functionnuclear receptor activity
D0006629biological_processlipid metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues20
DetailsBINDING SITE FOR RESIDUE 965 A 1500
ChainResidue
APHE268
AARG319
APHE329
ALEU330
APHE340
APHE349
AILE350
AILE353
APHE354
AHIS435
ALEU449
APHE271
ATRP457
ALEU274
AALA275
ASER278
AGLU281
AMET312
ALEU313
ATHR316

site_idAC2
Number of Residues16
DetailsBINDING SITE FOR RESIDUE 965 B 2500
ChainResidue
BHOH58
BSER242
BLEU274
BSER278
BMET312
BLEU313
BTHR316
BARG319
BPHE329
BLEU330
BPHE340
BPHE349
BILE353
BHIS435
BLEU449
BTRP457

site_idAC3
Number of Residues19
DetailsBINDING SITE FOR RESIDUE 965 D 3500
ChainResidue
DPHE271
DTHR272
DLEU274
DSER278
DGLU281
DILE309
DMET312
DLEU313
DTHR316
DARG319
DILE327
DPHE329
DLEU330
DPHE340
DPHE349
DILE353
DHIS435
DLEU449
DTRP457

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE IPA A 1501
ChainResidue
AGLN235
AGLU281
AILE282
APHE285
AGLU315

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE IPA B 2501
ChainResidue
BGLN235
BPHE285

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues11
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"20159957","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

250359

PDB entries from 2026-03-11

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