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1ISS

Crystal Structure of Metabotropic Glutamate Receptor Subtype 1 Complexed with an antagonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0004930molecular_functionG protein-coupled receptor activity
A0007186biological_processG protein-coupled receptor signaling pathway
A0016020cellular_componentmembrane
B0004930molecular_functionG protein-coupled receptor activity
B0007186biological_processG protein-coupled receptor signaling pathway
B0016020cellular_componentmembrane
Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MCG A 1001
ChainResidue
ATYR74
ASER165
ASER186
ATHR188
ALYS409

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MCG B 2001
ChainResidue
BTHR188
BTYR74
BTRP110
BSER165
BSER186

Functional Information from PROSITE/UniProt
site_idPS00979
Number of Residues19
DetailsG_PROTEIN_RECEP_F3_1 G-protein coupled receptors family 3 signature 1. VqNLLqLFdIPQIAySATS
ChainResidueDetails
AVAL171-SER189

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues10
DetailsBINDING: BINDING => ECO:0000269|PubMed:11069170, ECO:0000269|PubMed:11867751
ChainResidueDetails
ATYR74
BLYS409
ASER165
ATYR236
AASP318
ALYS409
BTYR74
BSER165
BTYR236
BASP318

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING:
ChainResidueDetails
ASER186
BSER186

site_idSWS_FT_FI3
Number of Residues4
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:11069170
ChainResidueDetails
AASN98
AASN223
BASN98
BASN223

site_idSWS_FT_FI4
Number of Residues4
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
AASN397
AASN515
BASN397
BASN515

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PDB entries from 2024-07-10

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