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9FZR

Wild-type EGFR in covalent complex with Poziotinib analogue

This is a non-PDB format compatible entry.
Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsDIAMOND BEAMLINE I03
Synchrotron siteDiamond
BeamlineI03
Temperature [K]100
Detector technologyPIXEL
Collection date2021-02-12
DetectorDECTRIS EIGER X 16M
Wavelength(s)0.898423
Spacegroup nameI 2 3
Unit cell lengths145.823, 145.823, 145.823
Unit cell angles90.00, 90.00, 90.00
Refinement procedure
Resolution59.603 - 1.991
Rwork0.186
R-free0.23320
Structure solution methodMOLECULAR REPLACEMENT
RMSD bond length0.008
RMSD bond angle1.723
Data reduction softwarexia2
Data scaling softwarepointless
Phasing softwarePHASER
Refinement softwareREFMAC (5.8.0430 (refmacat 0.4.82))
Data quality characteristics
 OverallOuter shell
Low resolution limit [Å]59.6032.040
High resolution limit [Å]1.9901.990
Rmerge0.1015.430
Number of reflections35412105527
<I/σ(I)>24
Completeness [%]100.0100
Redundancy41
CC(1/2)1.0000.396
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1VAPOR DIFFUSION, SITTING DROP829325mM TRIS-HCL pH8.0, 150mM NaCl, 5% Glycerol, 1mM TCEP, 100mM HEPES pH 7.4, 40% PEG400

239803

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