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3PPJ

Human B-Raf Kinase in Complex with a Furopyridine Inhibitor

Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeROTATING ANODE
Source detailsRIGAKU FR-E+ SUPERBRIGHT
Temperature [K]100
Detector technologyIMAGE PLATE
Collection date2005-07-15
DetectorRIGAKU RAXIS IV++
Wavelength(s)1.54
Spacegroup nameP 41 21 2
Unit cell lengths100.540, 100.540, 162.110
Unit cell angles90.00, 90.00, 90.00
Refinement procedure
Resolution27.480 - 3.700
R-factor0.251
Rwork0.250
R-free0.27200
Structure solution methodMOLECULAR REPLACEMENT
RMSD bond length0.007
RMSD bond angle1.100
Data reduction softwareMOSFLM
Data scaling softwareSCALA
Phasing softwareCNS
Refinement softwareCNS
Data quality characteristics
 OverallOuter shell
Low resolution limit [Å]30.0003.930
High resolution limit [Å]3.7003.700
Number of reflections9357
Completeness [%]100.0100
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1VAPOR DIFFUSION, HANGING DROP7293PEG 3350, pH 7.0, VAPOR DIFFUSION, HANGING DROP, temperature 293K

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