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2KSF
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BU of 2ksf by Molmil
Backbone structure of the membrane domain of E. coli histidine kinase receptor KdpD, Center for Structures of Membrane Proteins (CSMP) target 4312C
Descriptor: Sensor protein kdpD
Authors:Maslennikov, I, Klammt, C, Kefala, G, Okamura, M, Esquivies, L, Kwiatkowski, W, Choe, S, Center for Structures of Membrane Proteins (CSMP)
Deposit date:2010-01-03
Release date:2010-03-02
Last modified:2024-05-01
Method:SOLUTION NMR
Cite:Membrane domain structures of three classes of histidine kinase receptors by cell-free expression and rapid NMR analysis.
Proc.Natl.Acad.Sci.USA, 107, 2010
5AYF
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BU of 5ayf by Molmil
Crystal structure of SET7/9 in complex with cyproheptadine
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4-(dibenzo[1,2-a:2',1'-d][7]annulen-11-ylidene)-1-methyl-piperidine, Histone-lysine N-methyltransferase SETD7, ...
Authors:Niwa, H, Handa, N, Takemoto, Y, Ito, A, Tomabechi, Y, Umehara, T, Shirouzu, M, Yoshida, M, Yokoyama, S.
Deposit date:2015-08-20
Release date:2016-04-27
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.005 Å)
Cite:Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription
J.Med.Chem., 59, 2016
2KSD
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BU of 2ksd by Molmil
Backbone structure of the membrane domain of E. coli histidine kinase receptor ArcB, Center for Structures of Membrane Proteins (CSMP) target 4310C
Descriptor: Aerobic respiration control sensor protein arcB
Authors:Maslennikov, I, Klammt, C, Hwang, E, Kefala, G, Kwiatkowski, W, Jeon, Y, Choe, S, Center for Structures of Membrane Proteins (CSMP)
Deposit date:2010-01-02
Release date:2010-03-02
Last modified:2024-05-01
Method:SOLUTION NMR
Cite:Membrane domain structures of three classes of histidine kinase receptors by cell-free expression and rapid NMR analysis.
Proc.Natl.Acad.Sci.USA, 107, 2010
2KSE
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BU of 2kse by Molmil
Backbone structure of the membrane domain of E. coli histidine kinase receptor QseC, Center for Structures of Membrane Proteins (CSMP) target 4311C
Descriptor: Sensor protein qseC
Authors:Maslennikov, I, Klammt, C, Kefala, G, Esquivies, L, Kwiatkowski, W, Choe, S, Center for Structures of Membrane Proteins (CSMP)
Deposit date:2010-01-02
Release date:2010-03-02
Last modified:2024-05-01
Method:SOLUTION NMR
Cite:Membrane domain structures of three classes of histidine kinase receptors by cell-free expression and rapid NMR analysis.
Proc.Natl.Acad.Sci.USA, 107, 2010
8JOG
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BU of 8jog by Molmil
solution structure of Ras Binding Domein (RBD) in C-RAF with negative allosteric modulator.
Descriptor: RAF proto-oncogene serine/threonine-protein kinase
Authors:Makino, Y, Matsumoto, S, Yoshikawa, Y, Kawamura, T, Kumasaka, T, Shima, F.
Deposit date:2023-06-07
Release date:2024-06-12
Method:SOLUTION NMR
Cite:Small-molecule RAS/RAF-binding Inhibitors Allosterically Disrupt RAF Conformation and Exert Efficacy Against Broad-spectrum RAS-driven Cancers
To Be Published
8JOF
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BU of 8jof by Molmil
solution-structure of Ras Binding Domain (RBD) in C-RAF
Descriptor: RAF proto-oncogene serine/threonine-protein kinase
Authors:Makino, Y, Matsumoto, S, Yoshikawa, Y, Kawamura, T, Kumasaka, T, Shima, F.
Deposit date:2023-06-07
Release date:2024-06-12
Method:SOLUTION NMR
Cite:Small-molecule RAS/RAF-binding Inhibitors Allosterically Disrupt RAF Conformation and Exert Efficacy Against Broad-spectrum RAS-driven Cancers
To Be Published
8JNA
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BU of 8jna by Molmil
CRAF ras-binding domain chimera, apo form
Descriptor: RAF proto-oncogene serine/threonine-protein kinase, CRaf
Authors:Kawamura, T, Kumasaka, T.
Deposit date:2023-06-06
Release date:2024-06-19
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Small-molecule RAS/RAF-binding Inhibitors Allosterically Disrupt RAF Conformation and Exert Efficacy Against Broad-spectrum RAS-driven Cancers
To Be Published
8JNB
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BU of 8jnb by Molmil
CRAF ras-binding domain chimera, ligand complex
Descriptor: 2-[4-[[(2S)-1-ethanoyl-3-oxidanylidene-2H-indol-2-yl]methyl]-2-methoxy-phenoxy]ethanamide, RAF proto-oncogene serine/threonine-protein kinase, CRaf
Authors:Kawamura, T, Kumasaka, T.
Deposit date:2023-06-06
Release date:2024-06-19
Method:X-RAY DIFFRACTION (1.62 Å)
Cite:Small-molecule RAS/RAF-binding Inhibitors Allosterically Disrupt RAF Conformation and Exert Efficacy Against Broad-spectrum RAS-driven Cancers
To Be Published

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