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2ANP
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BU of 2anp by Molmil
Functional Glutamate 151 to Histidine mutant of the aminopeptidase from Aeromonas Proteolytica.
Descriptor: SODIUM ION, ZINC ION, leucyl aminopeptidase
Authors:Bzymek, K.P, Moulin, A, Swierczek, S.I, Ringe, D, Petsko, G.A, Holz, R.C.
Deposit date:2005-08-11
Release date:2005-10-04
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Kinetic, Spectroscopic, and X-ray Crystallographic Characterization of the Functional E151H Aminopeptidase from Aeromonas proteolytica.
Biochemistry, 44, 2005
3UEP
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BU of 3uep by Molmil
Crystal structure of YscQ-C from Yersinia pseudotuberculosis
Descriptor: YscQ-C, type III secretion protein
Authors:Bzymek, K.P, Ghosh, P.
Deposit date:2011-10-31
Release date:2012-04-04
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Two Translation Products of Yersinia yscQ Assemble To Form a Complex Essential to Type III Secretion.
Biochemistry, 51, 2012
4KAQ
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BU of 4kaq by Molmil
Structure of rituximab Fab
Descriptor: Rituximab heavy chain, Rituximab light chain
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2013-04-22
Release date:2014-12-24
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.48 Å)
Cite:Crystal structure of rituximab
To be Published
5ESQ
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BU of 5esq by Molmil
Cetuximab Fab in complex with cyclic beta-alanine-linked meditope
Descriptor: Cetuximab Fab heavy chain, Cetuximab Fab light chain, Cyclic beta-alanine-linked meditope, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2015-11-16
Release date:2016-06-15
Last modified:2017-12-13
Method:X-RAY DIFFRACTION (2.55 Å)
Cite:Cyclization strategies of meditopes: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5EUK
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BU of 5euk by Molmil
Cetuximab Fab in complex with F3H meditope variant
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cetuximab Fab heavy chain, Cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2015-11-18
Release date:2016-10-26
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5ETU
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BU of 5etu by Molmil
Cetuximab Fab in complex with L5E meditope variant
Descriptor: Cetuximab Fab heavy chain, Cetuximab Fab light chain, L5E meditope variant, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2015-11-18
Release date:2016-10-26
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.53 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5F88
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BU of 5f88 by Molmil
Cetuximab Fab in complex with L5Y meditope variant
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cetuximab Fab heavy chain, Cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2015-12-09
Release date:2016-10-26
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.481 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5FF6
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BU of 5ff6 by Molmil
Cetuximab Fab in complex with L10Q meditope variant
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cetuximab Fab heavy chain, Cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2015-12-17
Release date:2016-10-26
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
6AU5
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BU of 6au5 by Molmil
Structure of cetuximab with aminoheptanoic acid-linked n-butylarginine meditope variant
Descriptor: SULFATE ION, cetuximab Fab heavy chain, cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2017-08-30
Release date:2017-12-13
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.484 Å)
Cite:Meditope-Fab interaction: threading the hole.
Acta Crystallogr F Struct Biol Commun, 73, 2017
6AYN
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BU of 6ayn by Molmil
Structure of cetuximab with aminoheptanoic acid-linked N-(3-aminopropyl)-L-arginine meditope variant
Descriptor: Cetuximab Fab heavy chain, Cetuximab Fab light chain, Cyclic meditope
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2017-09-08
Release date:2017-12-13
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.48 Å)
Cite:Meditope-Fab interaction: threading the hole.
Acta Crystallogr F Struct Biol Commun, 73, 2017
6AZK
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BU of 6azk by Molmil
Structure of cetuximab with aminoheptanoic acid-linked N-(3-hydroxypropyl)-L-arginine meditope variant
Descriptor: SULFATE ION, cetuximab Fab heavy chain, cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2017-09-11
Release date:2017-12-13
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.477 Å)
Cite:Meditope-Fab interaction: threading the hole.
Acta Crystallogr F Struct Biol Commun, 73, 2017
6AXP
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BU of 6axp by Molmil
Structure of cetuximab with aminoheptanoic acid-linked n-octylarginine meditope variant
Descriptor: SULFATE ION, cetuximab Fab heavy chain, cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2017-09-07
Release date:2017-12-13
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.484 Å)
Cite:Meditope-Fab interaction: threading the hole.
Acta Crystallogr F Struct Biol Commun, 73, 2017
6AZL
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BU of 6azl by Molmil
Structure of cetuximab with aminoheptanoic acid-linked N-carboxyethylarginine meditope variant
Descriptor: SULFATE ION, cetuximab Fab heavy chain, cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2017-09-11
Release date:2017-12-13
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.482 Å)
Cite:Meditope-Fab interaction: threading the hole.
Acta Crystallogr F Struct Biol Commun, 73, 2017
5T1K
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BU of 5t1k by Molmil
Cetuximab Fab in complex with CQFDA(Ph)2STRRLKC
Descriptor: CETUXIMAB FAB HEAVY CHAIN, CETUXIMAB FAB LIGHT CHAIN, CQFDA(PH)2STRRLKC PEPTIDE, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-08-19
Release date:2016-10-26
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.48 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5T1M
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BU of 5t1m by Molmil
Cetuximab Fab in complex with CQYDLSTRRLKC
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CETUXIMAB FAB HEAVY CHAIN, CETUXIMAB FAB LIGHT CHAIN, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-08-19
Release date:2016-10-26
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.53 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5T1L
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BU of 5t1l by Molmil
Cetuximab Fab in complex with CQA(Ph)2DLSTRRLKC peptide
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CETUXIMAB FAB HEAVY CHAIN, CETUXIMAB FAB LIGHT CHAIN, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-08-19
Release date:2016-10-26
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.48 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5TH2
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BU of 5th2 by Molmil
Cetuximab Fab in complex with L5Q meditope variant
Descriptor: L5Q meditope, PHOSPHATE ION, cetuximab Fab, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-09-28
Release date:2016-10-26
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.84 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5U5F
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BU of 5u5f by Molmil
MEDITOPE ENABLED TRASTUZUMAB I83E VARIANT IN COMPLEX WITH (Ac) CQFDA(PH)2STRRLRCGGSK
Descriptor: 5-DIPHENYL LONG MEDITOPE, Immunoglobulin G binding protein A, MEMAB TRASTUZUMAB FAB HEAVY CHAIN, ...
Authors:Bzymek, K.P, Avery, K.N, Zer, C, Williams, J.C.
Deposit date:2016-12-06
Release date:2018-03-14
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.81 Å)
Cite:Meditope Enabled Trastuzumab I83E Variant In Complex With (Ac)Cqfda(Ph)2Strrlrcggsk
To Be Published
5U3D
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BU of 5u3d by Molmil
STRUCTURE OF MEDITOPE ENABLED TRASTUZUMAB I83E VARIANT
Descriptor: Immunoglobulin G binding protein A, MEMAB TRASTUZUMAB FAB HEAVY CHAIN, MEMAB TRASTUZUMAB FAB LIGHT CHAIN I83E, ...
Authors:Bzymek, K.P, Avery, K.N, Zer, C, Williams, J.C.
Deposit date:2016-12-01
Release date:2018-03-14
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.77 Å)
Cite:Meditope Enabled Trastuzumab I83E Variant
To Be Published
5HPM
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BU of 5hpm by Molmil
Cetuximab Fab in complex with cyclic linked meditope
Descriptor: 2-AMINO-3-MERCAPTO-PROPIONAMIDE, 2-acetamido-2-deoxy-beta-D-glucopyranose, Cetuximab Fab heavy chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-01-20
Release date:2016-06-15
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.67 Å)
Cite:Cyclization strategies of meditopes: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5HYQ
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BU of 5hyq by Molmil
Cetuximab Fab in complex with amidated meditope
Descriptor: Amidated meditope, Cetuximab heavy chain, Cetuximab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-02-01
Release date:2016-06-15
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.477 Å)
Cite:Cyclization strategies of meditopes: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5I2I
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BU of 5i2i by Molmil
Structure of cetuximab Fab with cyclic F3Q variant of the meditope
Descriptor: Cetuximab Fab heavy chain, Cetuximab Fab light chain, Meditope, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-02-08
Release date:2016-10-26
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.551 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5ICX
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BU of 5icx by Molmil
Cetuximab Fab in complex with CQFDLSTRRLRCGGSK meditope
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cetuximab Fab heavy chain, Cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-02-23
Release date:2016-06-15
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Cyclization strategies of meditopes: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5ID1
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BU of 5id1 by Molmil
Cetuximab Fab in complex with MPT-Cys meditope
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cetuximab Fab heavy chain, Cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-02-23
Release date:2016-06-15
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.49 Å)
Cite:Cyclization strategies of meditopes: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016
5IR1
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BU of 5ir1 by Molmil
Cetuximab Fab in complex with 3-bromophenylalanine meditope variant
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Cetuximab Fab heavy chain, Cetuximab Fab light chain, ...
Authors:Bzymek, K.P, Williams, J.C.
Deposit date:2016-03-11
Release date:2016-10-26
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.482 Å)
Cite:Natural and non-natural amino-acid side-chain substitutions: affinity and diffraction studies of meditope-Fab complexes.
Acta Crystallogr F Struct Biol Commun, 72, 2016

 

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