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3RIA
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BU of 3ria by Molmil
C. elegans glutamate-gated chloride channel (GluCl) in complex with Fab, ivermectin and iodide.
Descriptor: (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, Avermectin-sensitive glutamate-gated chloride channel GluCl alpha, CHLORIDE ION, ...
Authors:Hibbs, R.E, Gouaux, E.
Deposit date:2011-04-13
Release date:2011-05-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (3.8 Å)
Cite:Principles of activation and permeation in an anion-selective Cys-loop receptor.
Nature, 474, 2011
3RI5
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BU of 3ri5 by Molmil
C. elegans glutamate-gated chloride channel (GluCl) in complex with Fab, ivermectin and picrotoxin
Descriptor: (1aR,2aR,3S,6R,6aS,8aS,8bR,9R)-2a-hydroxy-8b-methyl-9-(prop-1-en-2-yl)hexahydro-3,6-methano-1,5,7-trioxacyclopenta[ij]c yclopropa[a]azulene-4,8(3H)-dione, (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Hibbs, R.E, Gouaux, E.
Deposit date:2011-04-12
Release date:2011-05-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (3.4 Å)
Cite:Principles of activation and permeation in an anion-selective Cys-loop receptor.
Nature, 474, 2011
3RHW
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BU of 3rhw by Molmil
C. elegans glutamate-gated chloride channel (GluCl) in complex with Fab and ivermectin
Descriptor: (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, 2-acetamido-2-deoxy-beta-D-glucopyranose, Avermectin-sensitive glutamate-gated chloride channel GluCl alpha, ...
Authors:Hibbs, R.E, Gouaux, E.
Deposit date:2011-04-12
Release date:2011-05-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (3.26 Å)
Cite:Principles of activation and permeation in an anion-selective Cys-loop receptor.
Nature, 474, 2011
3RIF
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BU of 3rif by Molmil
C. elegans glutamate-gated chloride channel (GluCl) in complex with Fab, ivermectin and glutamate.
Descriptor: (2aE,4E,5'S,6S,6'R,7S,8E,11R,13R,15S,17aR,20R,20aR,20bS)-6'-[(2S)-butan-2-yl]-20,20b-dihydroxy-5',6,8,19-tetramethyl-17 -oxo-3',4',5',6,6',10,11,14,15,17,17a,20,20a,20b-tetradecahydro-2H,7H-spiro[11,15-methanofuro[4,3,2-pq][2,6]benzodioxacy clooctadecine-13,2'-pyran]-7-yl 2,6-dideoxy-4-O-(2,6-dideoxy-3-O-methyl-alpha-L-arabino-hexopyranosyl)-3-O-methyl-alpha-L-arabino-hexopyranoside, 2-acetamido-2-deoxy-beta-D-glucopyranose, Avermectin-sensitive glutamate-gated chloride channel GluCl alpha, ...
Authors:Hibbs, R.E, Gouaux, E.
Deposit date:2011-04-13
Release date:2011-05-25
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (3.345 Å)
Cite:Principles of activation and permeation in an anion-selective Cys-loop receptor.
Nature, 474, 2011
4TNW
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BU of 4tnw by Molmil
C. elegans glutamate-gated chloride channel (GluCl) in complex with Fab and POPC in a lipid-modulated conformation
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, Avermectin-sensitive glutamate-gated chloride channel GluCl alpha, ...
Authors:Althoff, T, Hibbs, R.E, Banerjee, S, Gouaux, E.
Deposit date:2014-06-05
Release date:2014-08-13
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (3.2 Å)
Cite:X-ray structures of GluCl in apo states reveal a gating mechanism of Cys-loop receptors.
Nature, 512, 2014
4TNV
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BU of 4tnv by Molmil
C. elegans glutamate-gated chloride channel (GluCl) in complex with Fab in a non-conducting conformation
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Avermectin-sensitive glutamate-gated chloride channel GluCl alpha, CHLORIDE ION, ...
Authors:Althoff, T, Hibbs, R.E, Banerjee, S, Gouaux, E.
Deposit date:2014-06-05
Release date:2014-08-13
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (3.6 Å)
Cite:X-ray structures of GluCl in apo states reveal a gating mechanism of Cys-loop receptors.
Nature, 512, 2014
8DD3
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BU of 8dd3 by Molmil
Human GABAA receptor alpha1-beta2-gamma2 subtype in complex with GABA plus DMCM
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, GAMMA-AMINO-BUTANOIC ACID, ...
Authors:Zhu, S, Hibbs, R.E.
Deposit date:2022-06-17
Release date:2022-08-17
Last modified:2023-11-15
Method:ELECTRON MICROSCOPY (2.9 Å)
Cite:Structural and dynamic mechanisms of GABA A receptor modulators with opposing activities.
Nat Commun, 13, 2022
8DD2
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BU of 8dd2 by Molmil
Human GABAA receptor alpha1-beta2-gamma2 subtype in complex with GABA plus Zolpidem
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, GAMMA-AMINO-BUTANOIC ACID, ...
Authors:Zhu, S, Hibbs, R.E.
Deposit date:2022-06-17
Release date:2022-08-17
Last modified:2023-11-15
Method:ELECTRON MICROSCOPY (2.9 Å)
Cite:Structural and dynamic mechanisms of GABA A receptor modulators with opposing activities.
Nat Commun, 13, 2022
5KXI
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BU of 5kxi by Molmil
X-ray structure of the human Alpha4Beta2 nicotinic receptor
Descriptor: (S)-3-(1-METHYLPYRROLIDIN-2-YL)PYRIDINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, Neuronal acetylcholine receptor subunit alpha-4, ...
Authors:Morales-Perez, C.L, Noviello, C.M, Hibbs, R.E.
Deposit date:2016-07-20
Release date:2016-09-28
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.941 Å)
Cite:X-ray structure of the human alpha 4 beta 2 nicotinic receptor.
Nature, 538, 2016
8VRN
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BU of 8vrn by Molmil
Human GABAA receptor alpha1-beta2-gamma2 subtype in complex with GABA plus PPTQ
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3-(4-methylphenyl)-2-phenylquinazolin-4(3H)-one, ...
Authors:Chojnacka, W, Teng, J, Kim, J.J, Jensen, A.A, Hibbs, R.E.
Deposit date:2024-01-22
Release date:2024-06-26
Last modified:2024-07-03
Method:ELECTRON MICROSCOPY (2.57 Å)
Cite:Structural insights into GABA A receptor potentiation by Quaalude.
Nat Commun, 15, 2024
8VQY
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BU of 8vqy by Molmil
Human GABAA receptor alpha1-beta2-gamma2 subtype in complex with GABA plus methaqualone
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-methyl-3-(2-methylphenyl)quinazolin-4(3H)-one, GAMMA-AMINO-BUTANOIC ACID, ...
Authors:Chojnacka, W, Teng, J, Kim, J.J, Jensen, A.A, Hibbs, R.E.
Deposit date:2024-01-19
Release date:2024-06-26
Last modified:2024-07-03
Method:ELECTRON MICROSCOPY (2.82 Å)
Cite:Structural insights into GABA A receptor potentiation by Quaalude.
Nat Commun, 15, 2024
9AWK
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BU of 9awk by Molmil
Bovine fetal muscle nAChR resting state
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Li, H, Hibbs, R.E.
Deposit date:2024-03-05
Release date:2024-07-31
Last modified:2024-09-18
Method:ELECTRON MICROSCOPY (2.14 Å)
Cite:Structural switch in acetylcholine receptors in developing muscle.
Nature, 632, 2024
9AVU
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BU of 9avu by Molmil
Bovine fetal muscle nAChR bound to ACh
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINE, ...
Authors:Li, H, Hibbs, R.E.
Deposit date:2024-03-05
Release date:2024-07-31
Last modified:2024-09-18
Method:ELECTRON MICROSCOPY (2.45 Å)
Cite:Structural switch in acetylcholine receptors in developing muscle.
Nature, 632, 2024
9AVV
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BU of 9avv by Molmil
Bovine adult muscle nAChR resting state
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholine receptor subunit alpha, ...
Authors:Li, H, Hibbs, R.E.
Deposit date:2024-03-05
Release date:2024-07-31
Last modified:2024-09-18
Method:ELECTRON MICROSCOPY (2.09 Å)
Cite:Structural switch in acetylcholine receptors in developing muscle.
Nature, 632, 2024
9AWJ
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BU of 9awj by Molmil
Bovine adult muscle nAChR bound to ACh
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINE, ...
Authors:Li, H, Hibbs, R.E.
Deposit date:2024-03-05
Release date:2024-07-31
Last modified:2024-09-18
Method:ELECTRON MICROSCOPY (2.45 Å)
Cite:Structural switch in acetylcholine receptors in developing muscle.
Nature, 632, 2024
6UWZ
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BU of 6uwz by Molmil
Cryo-EM structure of Torpedo acetylcholine receptor in complex with alpha-bungarotoxin
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, Acetylcholine receptor subunit alpha, ...
Authors:Rahman, M.M, Teng, J, Worrell, B.T, Noveillo, C.M, Lee, M, Karlin, A, Stowell, M, Hibbs, R.E.
Deposit date:2019-11-06
Release date:2020-04-15
Last modified:2020-07-29
Method:ELECTRON MICROSCOPY (2.69 Å)
Cite:Structure of the Native Muscle-type Nicotinic Receptor and Inhibition by Snake Venom Toxins.
Neuron, 106, 2020
8EIZ
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BU of 8eiz by Molmil
Cryo-EM structure of squid sensory receptor CRB1
Descriptor: N-benzyl-2-(2,6-dimethylanilino)-N,N-diethyl-2-oxoethan-1-aminium, Squid sensory receptor CRB1, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose
Authors:Kang, G, Kim, J.J, Allard, C.A.H, Valencia-Montoya, W.A, van Giesen, L, Kilian, P.B, Bai, X, Bellono, N.W, Hibbs, R.E.
Deposit date:2022-09-15
Release date:2023-04-12
Last modified:2023-04-26
Method:ELECTRON MICROSCOPY (3.13 Å)
Cite:Sensory specializations drive octopus and squid behaviour.
Nature, 616, 2023
8EIS
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BU of 8eis by Molmil
Cryo-EM structure of octopus sensory receptor CRT1
Descriptor: 2-[2-[(1~{S},2~{S},4~{S},5'~{R},6~{R},7~{S},8~{R},9~{S},12~{S},13~{R},16~{S})-5',7,9,13-tetramethylspiro[5-oxapentacyclo[10.8.0.0^{2,9}.0^{4,8}.0^{13,18}]icos-18-ene-6,2'-oxane]-16-yl]oxyethyl]propane-1,3-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, Octopus sensory receptor
Authors:Kang, G, Kim, J.J, Allard, C.A.H, Valencia-Montoya, W.A, Bellono, N.W, Hibbs, R.E.
Deposit date:2022-09-15
Release date:2023-04-12
Last modified:2023-04-26
Method:ELECTRON MICROSCOPY (2.62 Å)
Cite:Sensory specializations drive octopus and squid behaviour.
Nature, 616, 2023
8F6Y
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BU of 8f6y by Molmil
Cryo-EM structure of Torpedo nicotinic acetylcholine receptor in complex with etomidate, desensitized-like state
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Goswami, U, Rahman, M.M, Teng, J, Hibbs, R.E.
Deposit date:2022-11-17
Release date:2023-06-07
Last modified:2024-01-31
Method:ELECTRON MICROSCOPY (2.79 Å)
Cite:Structural interplay of anesthetics and paralytics on muscle nicotinic receptors.
Nat Commun, 14, 2023
8ESK
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BU of 8esk by Molmil
Cryo-EM structure of Torpedo nicotinic acetylcholine receptor in complex with rocuronium, resting-like state
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Goswami, U, Rahman, M.M, Teng, J, Hibbs, R.E.
Deposit date:2022-10-14
Release date:2023-06-07
Last modified:2023-06-14
Method:ELECTRON MICROSCOPY (2.9 Å)
Cite:Structural interplay of anesthetics and paralytics on muscle nicotinic receptors.
Nat Commun, 14, 2023
8F6Z
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BU of 8f6z by Molmil
Cryo-EM structure of Torpedo nicotinic acetylcholine receptor in complex with succinylcholine, desensitized-like state
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2,2'-[(1,4-DIOXOBUTANE-1,4-DIYL)BIS(OXY)]BIS(N,N,N-TRIMETHYLETHANAMINIUM), 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Goswami, U, Rahman, M.M, Teng, J, Hibbs, R.E.
Deposit date:2022-11-17
Release date:2023-06-07
Last modified:2023-06-14
Method:ELECTRON MICROSCOPY (2.7 Å)
Cite:Structural interplay of anesthetics and paralytics on muscle nicotinic receptors.
Nat Commun, 14, 2023
8F2S
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BU of 8f2s by Molmil
Cryo-EM structure of Torpedo nicotinic acetylcholine receptor in complex with rocuronium, pore-blocked state
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Goswami, U, Rahman, M.M, Teng, J, Hibbs, R.E.
Deposit date:2022-11-08
Release date:2023-06-07
Last modified:2023-06-14
Method:ELECTRON MICROSCOPY (2.9 Å)
Cite:Structural interplay of anesthetics and paralytics on muscle nicotinic receptors.
Nat Commun, 14, 2023
6PV8
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BU of 6pv8 by Molmil
Human alpha3beta4 nicotinic acetylcholine receptor in complex with AT-1001
Descriptor: (3-endo)-N-(2-bromophenyl)-9-methyl-9-azabicyclo[3.3.1]nonan-3-amine, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Gharpure, A, Teng, J, Zhuang, Y, Noviello, C.M, Walsh, R.M, Cabuco, R, Howard, R.J, Zaveri, N.T, Lindahl, E, Hibbs, R.E.
Deposit date:2019-07-19
Release date:2019-09-11
Last modified:2020-07-29
Method:ELECTRON MICROSCOPY (3.87 Å)
Cite:Agonist Selectivity and Ion Permeation in the alpha 3 beta 4 Ganglionic Nicotinic Receptor.
Neuron, 104, 2019
6PV7
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BU of 6pv7 by Molmil
Human alpha3beta4 nicotinic acetylcholine receptor in complex with nicotine
Descriptor: (S)-3-(1-METHYLPYRROLIDIN-2-YL)PYRIDINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Gharpure, A, Teng, J, Zhuang, Y, Noviello, C.M, Walsh, R.M, Cabuco, R, Howard, R.J, Zaveri, N.T, Lindahl, E, Hibbs, R.E.
Deposit date:2019-07-19
Release date:2019-09-11
Last modified:2020-07-29
Method:ELECTRON MICROSCOPY (3.34 Å)
Cite:Agonist Selectivity and Ion Permeation in the alpha 3 beta 4 Ganglionic Nicotinic Receptor.
Neuron, 104, 2019
6PTZ
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BU of 6ptz by Molmil
Crystal structure of pigeon Cryptochrome 4 mutant Y319D in complex with flavin adenine dinucleotide
Descriptor: Cryptochrome-1, DI(HYDROXYETHYL)ETHER, FLAVIN-ADENINE DINUCLEOTIDE, ...
Authors:Zoltowski, B.D, Chelliah, Y, Wickramaratne, A.C, Jarocha, L, Karki, N, Mouritsen, H, Hore, P.J, Hibbs, R.E, Green, C.B, Takahashi, J.S.
Deposit date:2019-07-16
Release date:2019-09-04
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (1.793 Å)
Cite:Chemical and structural analysis of a photoactive vertebrate cryptochrome from pigeon.
Proc.Natl.Acad.Sci.USA, 116, 2019

 

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