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1CET
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CHLOROQUINE BINDS IN THE COFACTOR BINDING SITE OF PLASMODIUM FALCIPARUM LACTATE DEHYDROGENASE.
分子名称: N4-(7-CHLORO-QUINOLIN-4-YL)-N1,N1-DIETHYL-PENTANE-1,4-DIAMINE, PROTEIN (L-LACTATE DEHYDROGENASE)
著者Read, J.A, Wilkinson, K.W, Tranter, R, Sessions, R.B, Brady, R.L.
登録日1999-03-10
公開日1999-03-19
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Chloroquine binds in the cofactor binding site of Plasmodium falciparum lactate dehydrogenase.
J.Biol.Chem., 274, 1999
3LDH
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A comparison of the structures of apo dogfish m4 lactate dehydrogenase and its ternary complexes
分子名称: LACTATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, PYRUVIC ACID
著者White, J.L, Hackert, M.L, Buehner, M, Adams, M.J, Ford, G.C, Lentzjunior, P.J, Smiley, I.E, Steindel, S.J, Rossmann, M.G.
登録日1974-06-06
公開日1977-04-29
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献A comparison of the structures of apo dogfish M4 lactate dehydrogenase and its ternary complexes.
J.Mol.Biol., 102, 1976
1CIV
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CHLOROPLAST NADP-DEPENDENT MALATE DEHYDROGENASE FROM FLAVERIA BIDENTIS
分子名称: NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, NADP-MALATE DEHYDROGENASE
著者Carr, P.D, Ashton, A.R, Verger, D, Ollis, D.L.
登録日1999-04-01
公開日2000-04-05
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Chloroplast NADP-malate dehydrogenase: structural basis of light-dependent regulation of activity by thiol oxidation and reduction.
Structure Fold.Des., 7, 1999
1D3A
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BU of 1d3a by Molmil
CRYSTAL STRUCTURE OF THE WILD TYPE HALOPHILIC MALATE DEHYDROGENASE IN THE APO FORM
分子名称: CHLORIDE ION, HALOPHILIC MALATE DEHYDROGENASE, SODIUM ION
著者Richard, S.B, Madern, D, Garcin, E, Zaccai, G.
登録日1999-09-28
公開日2000-03-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.94 Å)
主引用文献Halophilic adaptation: novel solvent protein interactions observed in the 2.9 and 2.6 A resolution structures of the wild type and a mutant of malate dehydrogenase from Haloarcula marismortui.
Biochemistry, 39, 2000
1CEQ
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BU of 1ceq by Molmil
CHLOROQUINE BINDS IN THE COFACTOR BINDING SITE OF PLASMODIUM FALCIPARUM LACTATE DEHYDROGENASE.
分子名称: PROTEIN (L-LACTATE DEHYDROGENASE)
著者Read, J.A, Wilkinson, K.W, Tranter, R, Sessions, R.B, Brady, R.L.
登録日1999-03-10
公開日1999-03-19
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Chloroquine binds in the cofactor binding site of Plasmodium falciparum lactate dehydrogenase.
J.Biol.Chem., 274, 1999
5KKC
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l-lactate dehydrogenase from rabbit muscle with the inhibitor 6DHNAD
分子名称: L-lactate dehydrogenase A chain, SULFATE ION, [[(2~{R},3~{S},4~{R},5~{R})-5-(5-aminocarbonyl-2~{H}-pyridin-1-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methoxy-oxidanyl-phosphoryl] [(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl hydrogen phosphate
著者Meneely, K.M, Moran, G.R, Lamb, A.L.
登録日2016-06-21
公開日2016-11-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.859 Å)
主引用文献Ligand binding phenomena that pertain to the metabolic function of renalase.
Arch.Biochem.Biophys., 612, 2016
5KVV
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Structure of Malate Dehydrogenase in complex with NADH from Mycobacterium tuberculosis
分子名称: 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, ...
著者Cheng, Y.S, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC)
登録日2016-07-15
公開日2016-09-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Structure of Malate Dehydrogenase in complex with NADH from Mycobacterium tuberculosis
To Be Published
5KKA
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E. coli malate dehydrogenase with the inhibitor 6DHNAD
分子名称: Malate dehydrogenase, [[(2~{R},3~{S},4~{R},5~{R})-5-(5-aminocarbonyl-2~{H}-pyridin-1-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methoxy-oxidanyl-phosphoryl] [(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl hydrogen phosphate
著者Meneely, K.M, Lamb, A.L, Moran, G.R.
登録日2016-06-21
公開日2016-11-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Ligand binding phenomena that pertain to the metabolic function of renalase.
Arch.Biochem.Biophys., 612, 2016
1OC4
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Lactate dehydrogenase from Plasmodium berghei
分子名称: GLYCEROL, L-LACTATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Winter, V.J, Brady, R.L.
登録日2003-02-05
公開日2003-09-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of Plasmodium Berghei Lactate Dehydrogenase Indicates the Unique Structural Differences of These Enzymes are Shared Across the Plasmodium Genus
Mol.Biochem.Parasitol., 131, 2003
1O6Z
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1.95 A resolution structure of (R207S,R292S) mutant of malate dehydrogenase from the halophilic archaeon Haloarcula marismortui (holo form)
分子名称: CHLORIDE ION, MALATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Irimia, A, Ebel, C, Madern, D, Richard, S.B, Cosenza, L.W, Zaccai, G, Vellieux, F.M.D.
登録日2002-10-22
公開日2003-02-06
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The Oligomeric States of Haloarcula Marismortui Malate Dehydrogenase are Modulated by Solvent Components as Shown by Crystallographic and Biochemical Studies
J.Mol.Biol., 326, 2003
3NEP
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1.55A resolution structure of malate dehydrogenase from Salinibacter ruber
分子名称: Malate dehydrogenase
著者Coquelle, N, Madern, D.
登録日2010-06-09
公開日2010-10-13
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.551 Å)
主引用文献Gradual adaptive changes of a protein facing high salt concentrations.
J.Mol.Biol., 404, 2010
1EMD
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CRYSTAL STRUCTURE OF A TERNARY COMPLEX OF ESCHERICHIA COLI MALATE DEHYDROGENASE, CITRATE AND NAD AT 1.9 ANGSTROMS RESOLUTION
分子名称: CITRIC ACID, MALATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Hall, M.D, Banaszak, L.J.
登録日1993-03-25
公開日1993-10-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of a ternary complex of Escherichia coli malate dehydrogenase citrate and NAD at 1.9 A resolution.
J.Mol.Biol., 232, 1993
5LDH
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BU of 5ldh by Molmil
STRUCTURE OF THE ACTIVE TERNARY COMPLEX OF PIG HEART LACTATE DEHYDROGENASE WITH S-LAC-NAD AT 2.7 ANGSTROMS RESOLUTION
分子名称: (3S)-5-(3-CARBOXY-3-HYDROXYPROPYL) NICOTINAMIDE-ADENINE-DINUCLEOTIDE, CITRIC ACID, LACTATE DEHYDROGENASE
著者Grau, U.M, Rossmann, M.G.
登録日1980-10-29
公開日1981-03-04
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure of the active ternary complex of pig heart lactate dehydrogenase with S-lac-NAD at 2.7 A resolution.
J.Mol.Biol., 151, 1981
5UJK
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BU of 5ujk by Molmil
Malate dehydrogenase from Methylobacterium extorquens, complexed with NAD
分子名称: CALCIUM ION, CHLORIDE ION, Malate dehydrogenase, ...
著者Gonzalez, J.M.
登録日2017-01-18
公開日2017-02-08
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Conformational changes on substrate binding revealed by structures of Methylobacterium extorquens malate dehydrogenase.
Acta Crystallogr F Struct Biol Commun, 74, 2018
5MDH
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CRYSTAL STRUCTURE OF TERNARY COMPLEX OF PORCINE CYTOPLASMIC MALATE DEHYDROGENASE ALPHA-KETOMALONATE AND TNAD AT 2.4 ANGSTROMS RESOLUTION
分子名称: ALPHA-KETOMALONIC ACID, MALATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Chapman, A.D.M, Cortes, A, Dafforn, T.R, Clarke, A.R, Brady, R.L.
登録日1998-10-08
公開日1999-05-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis of substrate specificity in malate dehydrogenases: crystal structure of a ternary complex of porcine cytoplasmic malate dehydrogenase, alpha-ketomalonate and tetrahydoNAD.
J.Mol.Biol., 285, 1999
5ULV
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BU of 5ulv by Molmil
Malate dehydrogenase from Methylobacterium extorquens
分子名称: CALCIUM ION, Malate dehydrogenase
著者Gonzalez, J.M.
登録日2017-01-25
公開日2017-02-08
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.66 Å)
主引用文献Conformational changes on substrate binding revealed by structures of Methylobacterium extorquens malate dehydrogenase.
Acta Crystallogr F Struct Biol Commun, 74, 2018
1EZ4
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CRYSTAL STRUCTURE OF NON-ALLOSTERIC L-LACTATE DEHYDROGENASE FROM LACTOBACILLUS PENTOSUS AT 2.3 ANGSTROM RESOLUTION
分子名称: LACTATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Uchikoba, H, Fushinobu, S, Wakagi, T, Konno, M, Taguchi, H, Matsuzawa, H.
登録日2000-05-10
公開日2001-12-28
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of non-allosteric L-lactate dehydrogenase from Lactobacillus pentosus at 2.3 A resolution: specific interactions at subunit interfaces.
Proteins, 46, 2002
1PZH
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BU of 1pzh by Molmil
T.gondii LDH1 ternary complex with NAD and oxalate
分子名称: NICOTINAMIDE-ADENINE-DINUCLEOTIDE, OXALATE ION, lactate dehydrogenase
著者Kavanagh, K.L, Elling, R.A, Wilson, D.K.
登録日2003-07-10
公開日2004-02-24
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure of Toxoplasma gondii LDH1: Active-Site Differences from Human Lactate Dehydrogenases and the Structural Basis for Efficient APAD+ Use.
Biochemistry, 43, 2004
1PZE
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T.gondii LDH1 apo form
分子名称: lactate dehydrogenase
著者Kavanagh, K.L, Elling, R.A, Wilson, D.K.
登録日2003-07-10
公開日2004-02-24
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure of Toxoplasma gondii LDH1: Active-Site Differences from Human Lactate Dehydrogenases and the Structural Basis for Efficient APAD+ Use.
Biochemistry, 43, 2004
3P7M
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Structure of putative lactate dehydrogenase from Francisella tularensis subsp. tularensis SCHU S4
分子名称: Malate dehydrogenase, PHOSPHATE ION
著者Osinski, T, Cymborowski, M, Zimmerman, M.D, Gordon, E, Grimshaw, S, Skarina, T, Chruszcz, M, Savchenko, A, Anderson, W, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID)
登録日2010-10-12
公開日2010-10-20
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of putative lactate dehydrogenase from Francisella tularensis subsp. tularensis SCHU S4
To be Published
1PZF
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T.gondii LDH1 ternary complex with APAD+ and oxalate
分子名称: 3-ACETYLPYRIDINE ADENINE DINUCLEOTIDE, OXALATE ION, lactate dehydrogenase
著者Kavanagh, K.L, Elling, R.A, Wilson, D.K.
登録日2003-07-10
公開日2004-02-24
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of Toxoplasma gondii LDH1: Active-Site Differences from Human Lactate Dehydrogenases and the Structural Basis for Efficient APAD+ Use.
Biochemistry, 43, 2004
1PZG
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T.gondii LDH1 complexed with APAD and sulfate at 1.6 Angstroms
分子名称: 3-ACETYLPYRIDINE ADENINE DINUCLEOTIDE, SULFATE ION, lactate dehydrogenase
著者Kavanagh, K.L, Elling, R.A, Wilson, D.K.
登録日2003-07-10
公開日2004-02-24
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structure of Toxoplasma gondii LDH1: Active-Site Differences from Human Lactate Dehydrogenases and the Structural Basis for Efficient APAD+ Use.
Biochemistry, 43, 2004
3OM9
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T. Gondii bradyzoite-specific LDH (LDH1) in complex with NAD and OXQ
分子名称: 4-HYDROXY-1,2,5-OXADIAZOLE-3-CARBOXYLIC ACID, Lactate dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Susko, M.S, Wilson, D.K.
登録日2010-08-26
公開日2010-10-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献T.Gondii bradyzoite-specific LDH (LDH1) in complex with NAD and OXQ
To be Published
5NQB
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Rabbit Muscle L-lactate dehydrogenase in complex with malonate
分子名称: L-lactate dehydrogenase A chain, MALONATE ION
著者Luisi, B.F, Olin-Sandoval, V.
登録日2017-04-19
公開日2017-05-03
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献The self-inhibitory nature of metabolic networks and its alleviation through compartmentalization.
Nat Commun, 8, 2017
5NFR
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Crystal structure of malate dehydrogenase from Plasmodium falciparum (PfMDH)
分子名称: CITRIC ACID, Malate dehydrogenase
著者Lunev, S, Romero, A.R, Batista, F.A, Wrenger, C, Groves, M.R.
登録日2017-03-15
公開日2018-01-31
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Oligomeric interfaces as a tool in drug discovery: Specific interference with activity of malate dehydrogenase of Plasmodium falciparum in vitro.
PLoS ONE, 13, 2018

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