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2BZ4
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structure of E.coli KAS I H298Q mutant
分子名称: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE I, AMMONIUM ION, SULFATE ION
著者Olsen, J.G, von Wettstein-Knowles, P, Henriksen, A.
登録日2005-08-10
公開日2006-02-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Fatty acid synthesis. Role of active site histidines and lysine in Cys-His-His-type beta-ketoacyl-acyl carrier protein synthases.
FEBS J., 273, 2006
2C9H
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Structure of mitochondrial beta-ketoacyl synthase
分子名称: MITOCHONDRIAL BETA-KETOACYL SYNTHASE, NICKEL (II) ION
著者Bunkoczi, G, Wu, X, Smee, C, Gileadi, O, Arrowsmith, C, Edwards, A, Sundstrom, M, Weigelt, J, von Delft, F, Oppermann, U.
登録日2005-12-12
公開日2005-12-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure of Mitochondrial Beta-Ketoacyl Synthase
To be Published
2CDH
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ARCHITECTURE OF THE THERMOMYCES LANUGINOSUS FUNGAL FATTY ACID SYNTHASE AT 5 ANGSTROM RESOLUTION.
分子名称: DEHYDRATASE, ENOYL REDUCTASE, KETOACYL REDUCTASE, ...
著者Jenni, S, Leibundgut, M, Maier, T, Ban, N.
登録日2006-01-24
公開日2006-03-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (4.2 Å)
主引用文献Architecture of a Fungal Fatty Acid Synthase at 5 A Resolution.
Science, 311, 2006
2CF2
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Architecture of mammalian fatty acid synthase
分子名称: FATTY ACID SYNTHASE, DH DOMAIN, ER DOMAIN, ...
著者Maier, T, Jenni, S, Ban, N.
登録日2006-02-14
公開日2006-03-07
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (4.3 Å)
主引用文献Architecture of Mammalian Fatty Acid Synthase at 4.5 A Resolution.
Science, 311, 2006
2GFV
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Structure of E. coli FabF (KASII) C163Q mutant
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2
著者Soisson, S.M, Parthasarathy, G.
登録日2006-03-23
公開日2006-05-23
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献Platensimycin is a selective FabF inhibitor with potent antibiotic properties.
Nature, 441, 2006
2GFW
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Structure of wild type E. coli FabF (KASII)
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2
著者Soisson, S.M, Parthasarathy, G.
登録日2006-03-23
公開日2006-05-23
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Platensimycin is a selective FabF inhibitor with potent antibiotic properties.
Nature, 441, 2006
2GFX
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Structure of E. coli FabF(C163Q) in complex with Platensimycin
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2, PLATENSIMYCIN
著者Soisson, S.M, Parthasarathy, G.
登録日2006-03-23
公開日2006-05-23
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.59 Å)
主引用文献Platensimycin is a selective FabF inhibitor with potent antibiotic properties.
Nature, 441, 2006
2GFY
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Structure of E. coli FabF(K335A) mutant with covalently linked dodecanoic acid
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2, LAURIC ACID
著者Soisson, S.M, Parthasarathy, G.
登録日2006-03-23
公開日2006-05-23
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Platensimycin is a selective FabF inhibitor with potent antibiotic properties.
Nature, 441, 2006
2GP6
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X-ray crystal structure of Mycobacterium tuberculosis beta-ketoacyl acyl carrier protein synthase II (mtKasB)
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2
著者Sridharan, S, Sacchettini, J, TB Structural Genomics Consortium (TBSGC)
登録日2006-04-17
公開日2006-07-18
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献X-Ray Crystal Structure of Mycobacterium tuberculosis beta-Ketoacyl Acyl Carrier Protein Synthase II (mtKasB).
J.Mol.Biol., 366, 2007
2GQD
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The crystal structure of B-ketoacyl-ACP synthase II (FabF) from Staphylococcus aureus
分子名称: 3-oxoacyl-[acyl-carrier-protein] synthase 2
著者Miller, D.J, White, S.W, Zhang, Y.M, Rock, C.O.
登録日2006-04-20
公開日2006-05-02
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The crystal structure of B-ketoacyl-ACP synthase II (FabF) from Staphylococcus aureus
To be Published
2HG4
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Structure of the ketosynthase-acyltransferase didomain of module 5 from DEBS.
分子名称: 6-Deoxyerythronolide B Synthase, ACETATE ION, CHLORIDE ION, ...
著者Tang, Y, Kim, C.Y, Mathews, I.I, Cane, D.E, Khosla, C.
登録日2006-06-26
公開日2006-07-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.73 Å)
主引用文献The 2.7-A crystal structure of a 194-kDa homodimeric fragment of the 6-deoxyerythronolide B synthase.
Proc.Natl.Acad.Sci.Usa, 103, 2006
2IWY
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Human mitochondrial beta-ketoacyl ACP synthase
分子名称: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE, AMMONIUM ION
著者Christensen, C.E, Kragelund, B.B, von Wettstein-Knowles, P, Henriksen, A.
登録日2006-07-05
公開日2007-02-06
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Structure of the Human Beta-Ketoacyl [Acp] Synthase from the Mitochondrial Type II Fatty Acid Synthase.
Protein Sci., 16, 2007
2IWZ
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Human mitochondrial beta-ketoacyl ACP synthase complexed with hexanoic acid
分子名称: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE, AMMONIUM ION, HEXANOIC ACID
著者Christensen, C.E, Kragelund, B.B, von Wettstein-Knowles, P, Henriksen, A.
登録日2006-07-05
公開日2007-02-06
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structure of the Human Beta-Ketoacyl [Acp] Synthase from the Mitochondrial Type II Fatty Acid Synthase.
Protein Sci., 16, 2007
2IX4
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Arabidopsis thaliana mitochondrial beta-ketoacyl ACP synthase hexanoic acid complex
分子名称: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE, HEXANOIC ACID, POTASSIUM ION
著者Christensen, C.E, Kragelund, B.B, von Wettstein-Knowles, P, Henriksen, A.
登録日2006-07-06
公開日2007-02-06
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure of the Human Beta-Ketoacyl [Acp] Synthase from the Mitochondrial Type II Fatty Acid Synthase.
Protein Sci., 16, 2007
2PFF
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Structural Insights of Yeast Fatty Acid Synthase
分子名称: Fatty acid synthase subunit alpha, Fatty acid synthase subunit beta, Tail protein
著者Xiong, Y, Lomakin, I.B, Steitz, T.A.
登録日2007-04-04
公開日2007-07-10
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Structural Insights of Yeast Fatty Acid Synthase
Cell(Cambridge,Mass.), 129, 2007
2QO3
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Crystal Structure of [KS3][AT3] didomain from module 3 of 6-deoxyerthronolide B synthase
分子名称: (2S, 3R)-3-HYDROXY-4-OXO-7,10-TRANS,TRANS-DODECADIENAMIDE, ACETATE ION, ...
著者Khosla, C, Cane, E.D, Tang, Y, Chen, Y.A, Kim, C.Y.
登録日2007-07-19
公開日2007-09-04
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.59 Å)
主引用文献Structural and mechanistic analysis of protein interactions in module 3 of the 6-deoxyerythronolide B synthase
Chem.Biol., 14, 2007
2RJT
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Crystal Structure Analysis of a Surface Entropy Reduction Mutant of S. pneumoniae FabF
分子名称: Beta-ketoacyl-ACP synthase II
著者Soisson, S.M, Parthasarathy, G, Becker, J.
登録日2007-10-15
公開日2008-01-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Surface-entropy reduction approaches to manipulate crystal forms of beta-ketoacyl acyl carrier protein synthase II from Streptococcus pneumoniae.
Acta Crystallogr.,Sect.D, 64, 2008
2UV8
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Crystal structure of yeast fatty acid synthase with stalled acyl carrier protein at 3.1 angstrom resolution
分子名称: FATTY ACID SYNTHASE SUBUNIT ALPHA (FAS2), FATTY ACID SYNTHASE SUBUNIT BETA (FAS1), FLAVIN MONONUCLEOTIDE
著者Leibundgut, M, Jenni, S, Frick, C, Ban, N.
登録日2007-03-09
公開日2007-04-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural Basis for Substrate Delivery by Acyl Carrier Protein in the Yeast Fatty Acid Synthase
Science, 316, 2007
2VB7
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beta-ketoacyl-ACP synthase I (KAS) from E. coli, apo structure after soak in PEG solution
分子名称: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1
著者Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
登録日2007-09-06
公開日2007-12-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007
2VB8
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beta-ketoacyl-ACP synthase I (KAS) from E. coli with bound inhibitor thiolactomycin
分子名称: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1, CHLORIDE ION, THIOLACTOMYCIN
著者Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
登録日2007-09-06
公開日2007-12-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.52 Å)
主引用文献Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007
2VB9
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beta-ketoacyl-ACP synthase I (KAS) from E. coli, apo structure
分子名称: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1, CHLORIDE ION
著者Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
登録日2007-09-06
公開日2007-12-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007
2VBA
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beta-ketoacyl-ACP synthase I (KAS) from E. coli with bound amino- thiazole inhibitor
分子名称: 2-PHENYLAMINO-4-METHYL-5-ACETYL THIAZOLE, 3-OXOACYL-[ACYL-CARRIER-PROTEIN] SYNTHASE 1
著者Pappenberger, G, Schulz-Gasch, T, Bailly, J, Hennig, M.
登録日2007-09-06
公開日2007-12-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.36 Å)
主引用文献Structure-Assisted Discovery of an Aminothiazole Derivative as a Lead Molecule for Inhibition of Bacterial Fatty-Acid Synthesis.
Acta Crystallogr.,Sect.D, 63, 2007
2VKZ
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Structure of the cerulenin-inhibited fungal fatty acid synthase type I multienzyme complex
分子名称: (2S, 3R)-3-HYDROXY-4-OXO-7,10-TRANS,TRANS-DODECADIENAMIDE, FATTY ACID SYNTHASE SUBUNIT ALPHA, ...
著者Johansson, P, Wiltschi, B, Kumari, P, Kessler, B, Vonrhein, C, Vonck, J, Oesterhelt, D, Grininger, M.
登録日2008-01-07
公開日2008-08-12
最終更新日2017-06-21
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Inhibition of the Fungal Fatty Acid Synthase Type I Multienzyme Complex.
Proc.Natl.Acad.Sci.USA, 105, 2008
2VZ8
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Crystal Structure of Mammalian Fatty Acid Synthase
分子名称: FATTY ACID SYNTHASE
著者Maier, T, Leibundgut, M, Ban, N.
登録日2008-07-31
公開日2008-09-09
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.219 Å)
主引用文献The Crystal Structure of a Mammalian Fatty Acid Synthase.
Science, 321, 2008
2VZ9
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Crystal Structure of Mammalian Fatty Acid Synthase in complex with NADP
分子名称: FATTY ACID SYNTHASE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Maier, T, Leibundgut, M, Ban, N.
登録日2008-07-31
公開日2008-09-09
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献The Crystal Structure of a Mammalian Fatty Acid Synthase.
Science, 321, 2008

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