8F85
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![BU of 8f85 by Molmil](/molmil-images/mine/8f85) | |
8F84
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![BU of 8f84 by Molmil](/molmil-images/mine/8f84) | |
8F83
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![BU of 8f83 by Molmil](/molmil-images/mine/8f83) | |
8F82
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![BU of 8f82 by Molmil](/molmil-images/mine/8f82) | |
8F81
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![BU of 8f81 by Molmil](/molmil-images/mine/8f81) | |
8F80
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![BU of 8f80 by Molmil](/molmil-images/mine/8f80) | |
8F7Z
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![BU of 8f7z by Molmil](/molmil-images/mine/8f7z) | VRC34.01_mm28 bound to fusion peptide | Descriptor: | HIV-1 Env Fusion Peptide, VRC34_m228 Light Chain, VRC34_mm28 Heavy Chain | Authors: | Olia, A.S, Kwong, P.D. | Deposit date: | 2022-11-21 | Release date: | 2023-11-01 | Last modified: | 2024-02-14 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Antibody-directed evolution reveals a mechanism for enhanced neutralization at the HIV-1 fusion peptide site. Nat Commun, 14, 2023
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8F7V
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![BU of 8f7v by Molmil](/molmil-images/mine/8f7v) | Macrocyclic plasmin inhibitor | Descriptor: | (6S,9R,19S,22R)-N-{[4-(aminomethyl)phenyl]methyl}-22-[(benzenesulfonyl)amino]-3,12,21-trioxo-2,6,9,13,20-pentaazatetracyclo[22.2.2.2~6,9~.2~14,17~]dotriaconta-1(26),14,16,24,27,29-hexaene-19-carboxamide, GLYCEROL, Plasminogen, ... | Authors: | Guojie, W. | Deposit date: | 2022-11-20 | Release date: | 2023-02-08 | Last modified: | 2023-06-21 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | Synthesis and structural characterization of new macrocyclicplasmin inhibitors Chemmedchem, 2023
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8F7U
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![BU of 8f7u by Molmil](/molmil-images/mine/8f7u) | Macrocyclic Plasmin Inhibitor | Descriptor: | (5S,8R,18S,21R)-N-{[4-(aminomethyl)phenyl]methyl}-21-[(benzenesulfonyl)amino]-3,11,20-trioxo-2,5,8,12,19-pentaazatetracyclo[21.2.2.2~5,8~.2~13,16~]hentriaconta-1(25),13,15,23,26,28-hexaene-18-carboxamide, Activation peptide, GLYCEROL, ... | Authors: | Guojie, W. | Deposit date: | 2022-11-20 | Release date: | 2023-02-08 | Method: | X-RAY DIFFRACTION (1.47 Å) | Cite: | Synthesis and structural characterization of new macrocyclicplasmin inhibitors Chemmedchem, 2023
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8F7P
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![BU of 8f7p by Molmil](/molmil-images/mine/8f7p) | BRAF kinase in complex with LXH254 (naporafenib) | Descriptor: | N-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide, Serine/threonine-protein kinase B-raf | Authors: | Tkacik, E, Li, K, Gonzalez Del-Pino, G, Eck, M.J. | Deposit date: | 2022-11-20 | Release date: | 2023-04-12 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (2.74 Å) | Cite: | Structure and RAF family kinase isoform selectivity of type II RAF inhibitors tovorafenib and naporafenib. J.Biol.Chem., 299, 2023
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8F7O
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![BU of 8f7o by Molmil](/molmil-images/mine/8f7o) | BRAF kinase in complex with TAK580 (tovorafenib) | Descriptor: | 6-amino-5-chloro-N-[(1R)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide, Serine/threonine-protein kinase B-raf | Authors: | Tkacik, E, Li, K, Gonzalez Del-Pino, G, Eck, M.J. | Deposit date: | 2022-11-20 | Release date: | 2023-04-12 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (3.54 Å) | Cite: | Structure and RAF family kinase isoform selectivity of type II RAF inhibitors tovorafenib and naporafenib. J.Biol.Chem., 299, 2023
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8F7N
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![BU of 8f7n by Molmil](/molmil-images/mine/8f7n) | Crystal structure of chemoreceptor McpZ ligand sensing domain | Descriptor: | Methyl-accepting chemotaxis protein, YTTERBIUM (III) ION | Authors: | Salar, S, Schubot, F.D. | Deposit date: | 2022-11-19 | Release date: | 2023-07-05 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | The structural analysis of the periplasmic domain of Sinorhizobium meliloti chemoreceptor McpZ reveals a novel fold and suggests a complex mechanism of transmembrane signaling. Proteins, 91, 2023
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8F7K
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![BU of 8f7k by Molmil](/molmil-images/mine/8f7k) | Thermoplasma acidophilum 20S proteasome - wild type bound to ZYA | Descriptor: | N-[(benzyloxy)carbonyl]-L-tyrosyl-D-alanine, Proteasome subunit alpha, Proteasome subunit beta | Authors: | Chuah, J, Smith, D. | Deposit date: | 2022-11-18 | Release date: | 2023-08-30 | Method: | ELECTRON MICROSCOPY (1.94 Å) | Cite: | High resolution structures define divergent and convergent mechanisms of archaeal proteasome activation. Commun Biol, 6, 2023
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8F7I
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![BU of 8f7i by Molmil](/molmil-images/mine/8f7i) | The condensation domain of surfactin A synthetase C variant 18b in space group P43212 | Descriptor: | GLYCEROL, Surfactin synthetase | Authors: | Frota, N.F, Pistofidis, A, Folger, I.B, Hilvert, D, Schmeing, M. | Deposit date: | 2022-11-18 | Release date: | 2023-11-22 | Last modified: | 2024-06-12 | Method: | X-RAY DIFFRACTION (1.58 Å) | Cite: | High-throughput reprogramming of an NRPS condensation domain. Nat.Chem.Biol., 20, 2024
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8F7H
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![BU of 8f7h by Molmil](/molmil-images/mine/8f7h) | The condensation domain of surfactin A synthetase C variant 18b in space group P212121 | Descriptor: | GLYCEROL, Surfactin synthetase | Authors: | Frota, N.F, Pistofidis, A, Folger, I.B, Hilvert, D, Schmeing, M. | Deposit date: | 2022-11-18 | Release date: | 2023-11-22 | Last modified: | 2024-06-12 | Method: | X-RAY DIFFRACTION (1.93 Å) | Cite: | High-throughput reprogramming of an NRPS condensation domain. Nat.Chem.Biol., 20, 2024
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8F7G
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![BU of 8f7g by Molmil](/molmil-images/mine/8f7g) | The condensation domain of surfactin A synthetase C in space group P212121 | Descriptor: | GLYCEROL, Surfactin synthetase | Authors: | Frota, N.F, Pistofidis, A, Folger, I.B, Hilvert, D, Schmeing, T.M. | Deposit date: | 2022-11-18 | Release date: | 2023-11-22 | Last modified: | 2024-06-12 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | High-throughput reprogramming of an NRPS condensation domain. Nat.Chem.Biol., 20, 2024
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8F7F
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![BU of 8f7f by Molmil](/molmil-images/mine/8f7f) | The condensation domain of surfactin A synthetase C in space group P43212 | Descriptor: | GLYCEROL, Surfactin synthetase | Authors: | Frota, N, Pistofidis, A, Folger, I.B, Hilvert, D, Schmeing, T.M. | Deposit date: | 2022-11-18 | Release date: | 2023-11-22 | Last modified: | 2024-06-12 | Method: | X-RAY DIFFRACTION (1.62 Å) | Cite: | High-throughput reprogramming of an NRPS condensation domain. Nat.Chem.Biol., 20, 2024
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8F7C
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![BU of 8f7c by Molmil](/molmil-images/mine/8f7c) | Cryo-EM structure of human pannexin 2 | Descriptor: | Pannexin-2, Soluble cytochrome b562 fusion | Authors: | He, Z, Yuan, P. | Deposit date: | 2022-11-18 | Release date: | 2023-04-05 | Method: | ELECTRON MICROSCOPY (3.92 Å) | Cite: | Structural and functional analysis of human pannexin 2 channel. Nat Commun, 14, 2023
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8F76
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![BU of 8f76 by Molmil](/molmil-images/mine/8f76) | Human olfactory receptor OR51E2 bound to propionate in complex with miniGs399 | Descriptor: | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, Guanine nucleotide-binding protein G(s) subunit alpha isoforms short, ... | Authors: | Billesboelle, C.B, Manglik, A. | Deposit date: | 2022-11-18 | Release date: | 2023-03-22 | Last modified: | 2023-04-05 | Method: | ELECTRON MICROSCOPY (3.1 Å) | Cite: | Structural basis of odorant recognition by a human odorant receptor. Nature, 615, 2023
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8F70
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![BU of 8f70 by Molmil](/molmil-images/mine/8f70) | |
8F6V
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![BU of 8f6v by Molmil](/molmil-images/mine/8f6v) | |
8F6U
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![BU of 8f6u by Molmil](/molmil-images/mine/8f6u) | |
8F6P
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![BU of 8f6p by Molmil](/molmil-images/mine/8f6p) | Rat Cardiac Sodium Channel with Ranolazine Bound | Descriptor: | (R)-ranolazine, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | Authors: | Lenaeus, M.J, Tonggu, L. | Deposit date: | 2022-11-16 | Release date: | 2023-04-12 | Method: | ELECTRON MICROSCOPY (3.2 Å) | Cite: | Structural Basis for Inhibition of the Cardiac Sodium Channel by the Atypical Antiarrhythmic Drug Ranolazine To Be Published
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8F6O
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![BU of 8f6o by Molmil](/molmil-images/mine/8f6o) | anti-BTLA monoclonal antibody h22B3 in complex with BTLA | Descriptor: | B- and T-lymphocyte attenuator, h22B3 Fab heavy chain, h22B3 Fab light chain | Authors: | Hendle, J, Atwell, S, Lieu, R, Hickey, M, Weichert, K. | Deposit date: | 2022-11-16 | Release date: | 2023-05-24 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.31 Å) | Cite: | Epitope topography of agonist antibodies to the checkpoint inhibitory receptor BTLA. Structure, 31, 2023
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8F6N
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![BU of 8f6n by Molmil](/molmil-images/mine/8f6n) | Dihydropyrimidine Dehydrogenase (DPD) C671S Mutant Soaked with Thymine Quasi-Anaerobically | Descriptor: | Dihydropyrimidine dehydrogenase [NADP(+)], FLAVIN MONONUCLEOTIDE, FLAVIN-ADENINE DINUCLEOTIDE, ... | Authors: | Kaley, N, Smith, M, Forouzesh, D, Liu, D, Moran, G. | Deposit date: | 2022-11-16 | Release date: | 2023-02-01 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (2.12 Å) | Cite: | Mammalian dihydropyrimidine dehydrogenase: Added mechanistic details from transient-state analysis of charge transfer complexes. Arch.Biochem.Biophys., 736, 2023
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