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PDB: 5 results
2Y6O
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BU of 2y6o by Molmil
Crystal structure of EphA4 kinase domain in complex with Dasatinib.
Descriptor: EPHRIN TYPE-A RECEPTOR 4, N-(2-CHLORO-6-METHYLPHENYL)-2-({6-[4-(2-HYDROXYETHYL)PIPERAZIN-1-YL]-2-METHYLPYRIMIDIN-4-YL}AMINO)-1,3-THIAZOLE-5-CARBOXAMIDE
Authors:Farenc, C.J.A, Celie, P.H.N, Siegal, G.
Deposit date:2011-01-25
Release date:2011-11-02
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (1.543 Å)
Cite:Crystal Structure of the Epha4 Protein Tyrosine Kinase Domain in the Apo- and Dasatinib-Bound State.
FEBS Lett., 585, 2011
2Y6M
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BU of 2y6m by Molmil
Crystal structure of EphA4 kinase domain
Descriptor: EPHRIN TYPE-A RECEPTOR 4, GLYCEROL
Authors:Farenc, C.J.A, Celie, P.H.N, Siegal, G.
Deposit date:2011-01-25
Release date:2011-11-02
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Crystal Structure of the Epha4 Protein Tyrosine Kinase Domain in the Apo- and Dasatinib-Bound State.
FEBS Lett., 585, 2011
1B0X
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BU of 1b0x by Molmil
THE CRYSTAL STRUCTURE OF AN EPH RECEPTOR SAM DOMAIN REVEALS A MECHANISM FOR MODULAR DIMERIZATION.
Descriptor: PROTEIN (EPHA4 RECEPTOR TYROSINE KINASE)
Authors:Stapleton, D, Balan, I, Pawson, T, Sicheri, F.
Deposit date:1998-11-14
Release date:1999-05-03
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (2 Å)
Cite:The crystal structure of an Eph receptor SAM domain reveals a mechanism for modular dimerization.
Nat.Struct.Biol., 6, 1999
2XYU
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BU of 2xyu by Molmil
Crystal structure of EphA4 kinase domain in complex with VUF 12058
Descriptor: 5-(5-FLUORO-2-METHYLPHENYL)-6,7,8,9-TETRAHYDRO-3H-PYRAZOLO[3,4-C]ISOQUINOLIN-1-AMINE, EPHRIN TYPE-A RECEPTOR 4,, GLYCEROL
Authors:Farenc, C.J.A, Celie, P.H.N, vanLinden, O.P.J, Siegal, G.
Deposit date:2010-11-19
Release date:2011-11-30
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.117 Å)
Cite:Fragment Based Lead Discovery of Small Molecule Inhibitors for the Epha4 Receptor Tyrosine Kinase.
Eur.J.Med.Chem., 47, 2012
2HEL
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BU of 2hel by Molmil
Crystal structure of a mutant EphA4 kinase domain (Y742A)
Descriptor: Eph receptor A4
Authors:Wybenga-Groot, L.E, Sicheri, F, Pawson, T.
Deposit date:2006-06-21
Release date:2007-02-13
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:A change in conformational dynamics underlies the activation of Eph receptor tyrosine kinases.
EMBO J., 25, 2006

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