8SMC
| Cryo-EM structure of LRRK2 bound with type-I inhibitor DNL201 | Descriptor: | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1H-pyrazol-1-yl)propanenitrile, GUANOSINE-5'-DIPHOSPHATE, non-specific serine/threonine protein kinase | Authors: | Sun, J, Zhu, H. | Deposit date: | 2023-04-26 | Release date: | 2024-01-03 | Method: | ELECTRON MICROSCOPY (4.02 Å) | Cite: | Rab29-dependent asymmetrical activation of leucine-rich repeat kinase 2. Science, 382, 2023
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8FO2
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8FO9
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8FO8
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