Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 4 results

5C8Y
DownloadVisualize
BU of 5c8y by Molmil
Crystal structure of T2R-TTL-Plinabulin complex
Descriptor: (3Z,6Z)-3-benzylidene-6-[(5-tert-butyl-1H-imidazol-4-yl)methylidene]piperazine-2,5-dione, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Wang, Y, Yu, Y, Chen, Q, Yang, J.
Deposit date:2015-06-26
Release date:2015-11-04
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.594 Å)
Cite:Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery.
Febs J., 283, 2016
5CA1
DownloadVisualize
BU of 5ca1 by Molmil
Crystal structure of T2R-TTL-Nocodazole complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GLYCEROL, ...
Authors:Wang, Y, Yu, Y, Chen, Q, Yang, J.
Deposit date:2015-06-29
Release date:2015-11-04
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.401 Å)
Cite:Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery.
Febs J., 283, 2016
5CA0
DownloadVisualize
BU of 5ca0 by Molmil
Crystal structure of T2R-TTL-Lexibulin complex
Descriptor: 1-ethyl-3-[2-methoxy-4-(5-methyl-4-{[(1S)-1-(pyridin-3-yl)butyl]amino}pyrimidin-2-yl)phenyl]urea, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Wang, Y, Yu, Y, Chen, Q, Yang, J.
Deposit date:2015-06-29
Release date:2015-11-04
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.501 Å)
Cite:Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery.
Febs J., 283, 2016
5CB4
DownloadVisualize
BU of 5cb4 by Molmil
Crystal structure of T2R-TTL-Tivantinib complex
Descriptor: (3R,4R)-3-(5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-1-yl)-4-(1H-indol-3-yl)pyrrolidine-2,5-dione, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Wang, Y, Yu, Y, Chen, Q, Yang, J.
Deposit date:2015-06-30
Release date:2015-11-04
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.193 Å)
Cite:Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery.
Febs J., 283, 2016

218853

PDB entries from 2024-04-24

PDB statisticsPDBj update infoContact PDBjnumon