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PDB: 3 results

Crystal Structure of Falcipain-3 with Its inhibitor, K11017
Descriptor:	Cysteine protease falcipain-3, N~2~-(morpholin-4-ylcarbonyl)-N-[(3S)-1-phenyl-5-(phenylsulfonyl)pentan-3-yl]-L-leucinamide, SULFATE ION
Authors:	Kerr, I, Lee, J.H, Brinen, L.S.
Deposit date:	2008-01-09
Release date:	2009-01-20
Last modified:	2023-08-30
Method:	X-RAY DIFFRACTION (2.42 Å)
Cite:	Vinyl sulfones as antiparasitic agents and a structural basis for drug design. J.Biol.Chem., 284, 2009

Crystal structure analysis of cruzain bound to vinyl sulfone derived inhibitor (K11777)
Descriptor:	Cruzipain, NALPHA-[(4-METHYLPIPERAZIN-1-YL)CARBONYL]-N-{(1S)-3-PHENYL-1-[2-(PHENYLSULFONYL)ETHYL]PROPYL}-L-PHENYLALANINAMIDE, SULFATE ION
Authors:	Rickert, M, Brinen, L.
Deposit date:	2007-02-23
Release date:	2008-02-26
Last modified:	2019-09-04
Method:	X-RAY DIFFRACTION (1.95 Å)
Cite:	Vinyl sulfones as antiparasitic agents and a structural basis for drug design. J.Biol.Chem., 284, 2009

The crystal structure of rhodesain, the major cysteine protease of T. brucei rhodesiense, bound to inhibitor K777
Descriptor:	Cysteine protease, NALPHA-[(4-METHYLPIPERAZIN-1-YL)CARBONYL]-N-{(1S)-3-PHENYL-1-[2-(PHENYLSULFONYL)ETHYL]PROPYL}-L-PHENYLALANINAMIDE
Authors:	Brinen, L.S, Marion, R.
Deposit date:	2007-03-20
Release date:	2008-03-25
Last modified:	2023-08-30
Method:	X-RAY DIFFRACTION (1.65 Å)
Cite:	Vinyl sulfones as antiparasitic agents and a structural basis for drug design. J.Biol.Chem., 284, 2009