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PDB: 2 results

6KQQ
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BU of 6kqq by Molmil
NSD1 SET domain in complex with BT3 and SAM
Descriptor: 2-azanyl-6-[(2-azanyl-4-oxidanyl-1,3-benzothiazol-6-yl)disulfanyl]-1,3-benzothiazol-4-ol, 2-azanyl-6-sulfanyl-1,3-benzothiazol-4-ol, CALCIUM ION, ...
Authors:Cho, H.J, Cierpicki, T.
Deposit date:2019-08-18
Release date:2020-09-02
Last modified:2022-03-23
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Covalent inhibition of NSD1 histone methyltransferase.
Nat.Chem.Biol., 16, 2020
6KQP
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BU of 6kqp by Molmil
NSD1 SET domain in complex with SAM
Descriptor: Histone-lysine N-methyltransferase, H3 lysine-36 and H4 lysine-20 specific, S-ADENOSYLMETHIONINE, ...
Authors:Cho, H.J, Cierpicki, T.
Deposit date:2019-08-18
Release date:2020-09-02
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Covalent inhibition of NSD1 histone methyltransferase.
Nat.Chem.Biol., 16, 2020

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