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PDB: 3 results

4HCO
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BU of 4hco by Molmil
Human Plk1-PBD in complex with Thymoquinone at the phophopeptide binding site
Descriptor: 2-methyl-5-(1-methylethyl)cyclohexa-2,5-diene-1,4-dione, GLYCEROL, Serine/threonine-protein kinase PLK1
Authors:Yin, Z, Rehse, P.H.
Deposit date:2012-10-01
Release date:2012-10-10
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.75 Å)
Cite:Thymoquinone Blocks pSer/pThr Recognition by Plk1 Polo-Box Domain As a Phosphate Mimic
Acs Chem.Biol., 8, 2013
4H5X
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BU of 4h5x by Molmil
human Plk1-PBD with a glycerol bound at the phophopeptide binding site
Descriptor: GLYCEROL, Serine/threonine-protein kinase PLK1
Authors:Yin, Z, Rehse, P.H.
Deposit date:2012-09-19
Release date:2012-10-03
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Thymoquinone Blocks pSer/pThr Recognition by Plk1 Polo-Box Domain As a Phosphate Mimic
Acs Chem.Biol., 8, 2013
4H71
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BU of 4h71 by Molmil
Human Plk1-PBD in complex with Poloxime ((E)-4-(hydroxyimino)-2-isopropyl-5-methylcyclohexa-2,5-dienone)
Descriptor: 2-methyl-5-(1-methylethyl)cyclohexa-2,5-diene-1,4-dione 1-oxime, GLYCEROL, Serine/threonine-protein kinase PLK1
Authors:Yin, Z, Rehse, P.H.
Deposit date:2012-09-19
Release date:2012-10-03
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.93 Å)
Cite:Thymoquinone Blocks pSer/pThr Recognition by Plk1 Polo-Box Domain As a Phosphate Mimic
Acs Chem.Biol., 8, 2013

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PDB entries from 2024-05-01

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