4H71
Human Plk1-PBD in complex with Poloxime ((E)-4-(hydroxyimino)-2-isopropyl-5-methylcyclohexa-2,5-dienone)
Replaces: 3MHNSummary for 4H71
Entry DOI | 10.2210/pdb4h71/pdb |
Related | 4H5X 4H70 |
Descriptor | Serine/threonine-protein kinase PLK1, GLYCEROL, 2-methyl-5-(1-methylethyl)cyclohexa-2,5-diene-1,4-dione 1-oxime, ... (4 entities in total) |
Functional Keywords | kinase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: P53350 |
Total number of polymer chains | 2 |
Total formula weight | 55360.06 |
Authors | Yin, Z.,Rehse, P.H. (deposition date: 2012-09-19, release date: 2012-10-03, Last modification date: 2023-11-08) |
Primary citation | Yin, Z.,Song, Y.,Rehse, P.H. Thymoquinone Blocks pSer/pThr Recognition by Plk1 Polo-Box Domain As a Phosphate Mimic Acs Chem.Biol., 8:303-308, 2013 Cited by PubMed: 23135290DOI: 10.1021/cb3004379 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.93 Å) |
Structure validation
Download full validation report