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PDB: 3 results

8B5B
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BU of 8b5b by Molmil
Human BRD4 bromdomain 1 in complex with a H4 peptide containing acetyl lysine and ApmTri (H4K5acK8ApmTri)
Descriptor: Bromodomain-containing protein 4, DI(HYDROXYETHYL)ETHER, H4K5acK8ApmTri
Authors:Braun, M.B, Bartlick, N, Stehle, T.
Deposit date:2022-09-22
Release date:2023-01-11
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.92 Å)
Cite:Synthesis, Biochemical Characterization, and Genetic Encoding of a 1,2,4-Triazole Amino Acid as an Acetyllysine Mimic for Bromodomains of the BET Family.
Angew.Chem.Int.Ed.Engl., 62, 2023
8B5C
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BU of 8b5c by Molmil
Human BRD4 bromdomain 1 in complex with a H4 peptide containing ApmTri (H4K5/8ApmTri)
Descriptor: Bromodomain-containing protein 4, H4K5/8ApmTri
Authors:Braun, M.B, Bartlick, N, Stehle, T.
Deposit date:2022-09-22
Release date:2023-01-11
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.58 Å)
Cite:Synthesis, Biochemical Characterization, and Genetic Encoding of a 1,2,4-Triazole Amino Acid as an Acetyllysine Mimic for Bromodomains of the BET Family.
Angew.Chem.Int.Ed.Engl., 62, 2023
8B5A
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BU of 8b5a by Molmil
Human BRD3 bromodomain 2 in complex with a H4 peptide containing ApmTri (H4K20ApmTri)
Descriptor: Bromodomain-containing protein 3, H4K20ApmTri
Authors:Braun, M.B, Bartlick, N, Stehle, T.
Deposit date:2022-09-22
Release date:2023-01-11
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.92 Å)
Cite:Synthesis, Biochemical Characterization, and Genetic Encoding of a 1,2,4-Triazole Amino Acid as an Acetyllysine Mimic for Bromodomains of the BET Family.
Angew.Chem.Int.Ed.Engl., 62, 2023

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PDB entries from 2024-07-10

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