7D6F
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![BU of 7d6f by Molmil](/molmil-images/mine/7d6f) | The crystal structure of ARMS-PBM/MAGI2-PDZ4 | Descriptor: | GLYCEROL, Kinase D-interacting substrate of 220 kDa, Membrane-associated guanylate kinase, ... | Authors: | Ye, J, Zhang, Y, Zhong, Z, Wang, C. | Deposit date: | 2020-09-30 | Release date: | 2020-11-04 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (3.001 Å) | Cite: | Crystal structure of the PDZ4 domain of MAGI2 in complex with PBM of ARMS reveals a canonical PDZ recognition mode. Neurochem.Int., 149, 2021
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6LCB
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![BU of 6lcb by Molmil](/molmil-images/mine/6lcb) | Crystal structure of human Dishevelled1 PDZ domain with its inhibitor NPL3009 | Descriptor: | 2-[[3-[(2E)-2-[1,3-bis(oxidanylidene)-1-phenyl-butan-2-ylidene]hydrazinyl]phenyl]sulfonylamino]benzoic acid, SULFATE ION, Segment polarity protein dishevelled homolog DVL-1 | Authors: | Yasukochi, S, Numoto, N, Tenno, N, Tenno, T, Ito, N, Hiroaki, H. | Deposit date: | 2019-11-18 | Release date: | 2020-11-25 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.4 Å) | Cite: | Crystal structure of human Dishevelled1 PDZ domain with its inhibitor NPL3009 To Be Published
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6LCA
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![BU of 6lca by Molmil](/molmil-images/mine/6lca) | Crystal structure of human Dishevelled1 PDZ domain homotrimer | Descriptor: | SULFATE ION, Segment polarity protein dishevelled homolog DVL-1 | Authors: | Yasukochi, S, Numoto, N, Tenno, N, Tenno, T, Ito, N, Hiroaki, H. | Deposit date: | 2019-11-18 | Release date: | 2020-11-25 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Crystal structure of human Dishevelled1 PDZ domain homotrimer To Be Published
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6X1N
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![BU of 6x1n by Molmil](/molmil-images/mine/6x1n) | |
6X20
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![BU of 6x20 by Molmil](/molmil-images/mine/6x20) | |
6X22
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![BU of 6x22 by Molmil](/molmil-images/mine/6x22) | |
6X1X
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![BU of 6x1x by Molmil](/molmil-images/mine/6x1x) | PDZ domain from choanoflagellate GIPC (mbGIPC) | Descriptor: | GLYCEROL, mbGIPC protein | Authors: | Gao, M, Amacher, J.F. | Deposit date: | 2020-05-19 | Release date: | 2020-11-25 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (1.198 Å) | Cite: | Structural characterization and computational analysis of PDZ domains in Monosiga brevicollis. Protein Sci., 29, 2020
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6X23
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![BU of 6x23 by Molmil](/molmil-images/mine/6x23) | |
6X1P
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![BU of 6x1p by Molmil](/molmil-images/mine/6x1p) | |
6X1R
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![BU of 6x1r by Molmil](/molmil-images/mine/6x1r) | |
7CQF
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![BU of 7cqf by Molmil](/molmil-images/mine/7cqf) | |
6T36
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![BU of 6t36 by Molmil](/molmil-images/mine/6t36) | Crystal structure of the PTPN3 PDZ domain bound to the HBV core protein C-terminal peptide | Descriptor: | BROMIDE ION, Capsid protein, Tyrosine-protein phosphatase non-receptor type 3 | Authors: | Genera, M, Mechaly, A, Haouz, A, Caillet-Saguy, C. | Deposit date: | 2019-10-10 | Release date: | 2021-01-20 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.86 Å) | Cite: | Molecular basis of the interaction of the human tyrosine phosphatase PTPN3 with the hepatitis B virus core protein. Sci Rep, 11, 2021
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6RLC
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![BU of 6rlc by Molmil](/molmil-images/mine/6rlc) | Crystal structure of the PDZ tandem of syntenin in complex with fragment F13 | Descriptor: | (2~{S})-2-[3-(4-chlorophenyl)sulfanylpropanoylamino]-3-methyl-butanoic acid, ACETATE ION, Syntenin-1 | Authors: | Feracci, M, Barral, K. | Deposit date: | 2019-05-02 | Release date: | 2021-02-03 | Last modified: | 2024-05-15 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loadifing with syndecan and EpCAM cargo. J Extracell Vesicles, 10, 2020
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6R9H
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![BU of 6r9h by Molmil](/molmil-images/mine/6r9h) | Crystal structure of the PDZ tandem of syntenin in complex with fragment C58 | Descriptor: | (2~{S})-2-[2-(4-chlorophenyl)sulfanylethanoylamino]-3-methyl-butanoic acid, ACETATE ION, PHOSPHATE ION, ... | Authors: | Feracci, M, Barral, K. | Deposit date: | 2019-04-03 | Release date: | 2021-02-03 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loadifing with syndecan and EpCAM cargo. J Extracell Vesicles, 10, 2020
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6V84
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![BU of 6v84 by Molmil](/molmil-images/mine/6v84) | |
6XA8
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![BU of 6xa8 by Molmil](/molmil-images/mine/6xa8) | |
6XA6
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![BU of 6xa6 by Molmil](/molmil-images/mine/6xa6) | |
6XA7
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![BU of 6xa7 by Molmil](/molmil-images/mine/6xa7) | |
7JO7
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![BU of 7jo7 by Molmil](/molmil-images/mine/7jo7) | Crystal Structure of Human Scribble PDZ2 | Descriptor: | 1,2-ETHANEDIOL, Protein scribble homolog | Authors: | How, J.Y, Kvansakul, M. | Deposit date: | 2020-08-06 | Release date: | 2021-03-24 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.44 Å) | Cite: | Structural basis of the human Scribble-Vangl2 association in health and disease. Biochem.J., 478, 2021
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7M4R
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![BU of 7m4r by Molmil](/molmil-images/mine/7m4r) | |
7NTJ
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![BU of 7ntj by Molmil](/molmil-images/mine/7ntj) | PALS1 PDZ1 domain with SARS-CoV-1_E PBM complex | Descriptor: | Envelope small membrane protein, MAGUK p55 subfamily member 5 | Authors: | Javorsky, A, Kvansakul, M. | Deposit date: | 2021-03-10 | Release date: | 2021-06-16 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.74 Å) | Cite: | Structural basis of coronavirus E protein interactions with human PALS1 PDZ domain. Commun Biol, 4, 2021
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7NTK
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![BU of 7ntk by Molmil](/molmil-images/mine/7ntk) | PALS1 PDZ1 domain with SARS-CoV-2_E PBM complex | Descriptor: | 1,2-ETHANEDIOL, CITRATE ANION, Envelope small membrane protein, ... | Authors: | Javorsky, A, Kvansakul, M. | Deposit date: | 2021-03-10 | Release date: | 2021-06-16 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Structural basis of coronavirus E protein interactions with human PALS1 PDZ domain. Commun Biol, 4, 2021
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6ZBQ
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![BU of 6zbq by Molmil](/molmil-images/mine/6zbq) | Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling | Descriptor: | 5-fluoranyl-2-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonylamino)benzoic acid, Dishevelled, dsh homolog 3 (Drosophila), ... | Authors: | Roske, Y, Heinemann, U, Oschkinat, H. | Deposit date: | 2020-06-09 | Release date: | 2021-06-23 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.43 Å) | Cite: | Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling J.Magn.Reson., 2021
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6ZBZ
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![BU of 6zbz by Molmil](/molmil-images/mine/6zbz) | Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling | Descriptor: | 1,2-ETHANEDIOL, 2-[(3,4-dimethylphenyl)sulfonylamino]-5-fluoranyl-benzoic acid, Dishevelled, ... | Authors: | Roske, Y, Heinemann, U, Oschkinat, H. | Deposit date: | 2020-06-09 | Release date: | 2021-06-23 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling J.Magn.Reson., 2021
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6ZC7
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![BU of 6zc7 by Molmil](/molmil-images/mine/6zc7) | |