1F57
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![BU of 1f57 by Molmil](/molmil-images/mine/1f57) | |
8CPA
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![BU of 8cpa by Molmil](/molmil-images/mine/8cpa) | |
4F8Z
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![BU of 4f8z by Molmil](/molmil-images/mine/4f8z) | Carboxypeptidase T with Boc-Leu | Descriptor: | CALCIUM ION, Carboxypeptidase T, GLYCEROL, ... | Authors: | Timofeev, V.I, Kuznetsov, S.A, Akparov, V.K, Kuranova, I.P. | Deposit date: | 2012-05-18 | Release date: | 2013-05-22 | Last modified: | 2015-09-30 | Method: | X-RAY DIFFRACTION (1.38 Å) | Cite: | Three-dimensional structure of carboxypeptidase T from Thermoactinomyces vulgaris in complex with N-BOC-L-leucine. Biochemistry Mosc., 78, 2013
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7Q87
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![BU of 7q87 by Molmil](/molmil-images/mine/7q87) | Carboxypeptidase T with (S)-3-phenyllactic acid | Descriptor: | ALPHA-HYDROXY-BETA-PHENYL-PROPIONIC ACID, CALCIUM ION, Carboxypeptidase T, ... | Authors: | Timofeev, V.I, Akparov, V.K, Shevtsov, M.B, Kuranova, I.P. | Deposit date: | 2021-11-10 | Release date: | 2022-01-26 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (1.73 Å) | Cite: | Carboxypeptidase T with (S)-3-phenyllactic acid To Be Published
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2JEW
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![BU of 2jew by Molmil](/molmil-images/mine/2jew) | |
4Z65
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![BU of 4z65 by Molmil](/molmil-images/mine/4z65) | Carboxypeptidase B with Sulphamoil Arginine | Descriptor: | Carboxypeptidase B, N~2~-sulfamoyl-L-arginine, ZINC ION | Authors: | Timofeev, V.I, Akparov, V.K, Kuranova, I.P. | Deposit date: | 2015-04-03 | Release date: | 2015-10-14 | Last modified: | 2015-10-28 | Method: | X-RAY DIFFRACTION (1.25 Å) | Cite: | Structure of the complex of carboxypeptidase B and N-sulfamoyl-L-arginine. Acta Crystallogr.,Sect.F, 71, 2015
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6Z28
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![BU of 6z28 by Molmil](/molmil-images/mine/6z28) | |
5ZEQ
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![BU of 5zeq by Molmil](/molmil-images/mine/5zeq) | Carboxypeptidase B in complex with DD28 | Descriptor: | (2~{S})-2-[(6-azanyl-5-chloranyl-pyridin-3-yl)methyl]-3-selanyl-propanoic acid, CACODYLATE ION, Carboxypeptidase B, ... | Authors: | Itoh, T, Yoshimoto, N, Yamamoto, K. | Deposit date: | 2018-02-27 | Release date: | 2018-06-20 | Last modified: | 2018-07-04 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Structural basis for the selective inhibition of activated thrombin-activatable fibrinolysis inhibitor (TAFIa) by a selenium-containing inhibitor with chloro-aminopyridine as a basic group Bioorg. Med. Chem. Lett., 28, 2018
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6I6Z
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![BU of 6i6z by Molmil](/molmil-images/mine/6i6z) | |
8QVO
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![BU of 8qvo by Molmil](/molmil-images/mine/8qvo) | L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris | Descriptor: | CALCIUM ION, Carboxypeptidase T, SULFATE ION, ... | Authors: | Timofeev, V.I, Dorovatovskii, P.V, Lazarenko, V.A, Akparov, V.K, Kuranova, I.P. | Deposit date: | 2023-10-18 | Release date: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.96 Å) | Cite: | L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris To Be Published
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6CPA
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![BU of 6cpa by Molmil](/molmil-images/mine/6cpa) | |
5CPA
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![BU of 5cpa by Molmil](/molmil-images/mine/5cpa) | |
2RFH
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![BU of 2rfh by Molmil](/molmil-images/mine/2rfh) | |
5J1Q
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![BU of 5j1q by Molmil](/molmil-images/mine/5j1q) | |
5JC6
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![BU of 5jc6 by Molmil](/molmil-images/mine/5jc6) | |
4OKO
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![BU of 4oko by Molmil](/molmil-images/mine/4oko) | Crystal structure of Francisella tularensis REP34 (Rapid Encystment Phenotype Protein 34 KDa) | Descriptor: | ACETATE ION, Rapid Encystment Phenotype Protein 34 KDa, ZINC ION | Authors: | Feld, G.K, Segelke, B.W, Corzett, M.H, Hunter, M.S, Frank, M, Rasley, A. | Deposit date: | 2014-01-22 | Release date: | 2014-09-24 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.053 Å) | Cite: | Structure and Function of REP34 Implicates Carboxypeptidase Activity in Francisella tularensis Host Cell Invasion. J.Biol.Chem., 289, 2014
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7AQP
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![BU of 7aqp by Molmil](/molmil-images/mine/7aqp) | T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris | Descriptor: | CALCIUM ION, Carboxypeptidase T, SULFATE ION, ... | Authors: | Timofeev, V.I, Akparov, V.K, Kuranova, I.P. | Deposit date: | 2020-10-22 | Release date: | 2020-12-02 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris To Be Published
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7ARU
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![BU of 7aru by Molmil](/molmil-images/mine/7aru) | |
2V77
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![BU of 2v77 by Molmil](/molmil-images/mine/2v77) | Crystal Structure of Human Carboxypeptidase A1 | Descriptor: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CARBOXYPEPTIDASE A1, OCTANE-1,3,5,7-TETRACARBOXYLIC ACID, ... | Authors: | Pallares, I, Fernandez, D, Comellas-Bigler, M, Fernandez-Recio, J, Ventura, S, Aviles, F.X, Vendrell, J. | Deposit date: | 2007-07-27 | Release date: | 2008-07-01 | Last modified: | 2023-12-13 | Method: | X-RAY DIFFRACTION (1.603 Å) | Cite: | Direct interaction between a human digestive protease and the mucoadhesive poly(acrylic acid). Acta Crystallogr. D Biol. Crystallogr., D64, 2008
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3PRT
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![BU of 3prt by Molmil](/molmil-images/mine/3prt) | Mutant of the Carboxypeptidase T | Descriptor: | CALCIUM ION, Carboxypeptidase T, GLYCEROL, ... | Authors: | Timofeev, V.I, Akparov, V.K, Grishin, A.M, Kuranova, I.P. | Deposit date: | 2010-11-30 | Release date: | 2011-11-30 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (1.66 Å) | Cite: |
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3QNV
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![BU of 3qnv by Molmil](/molmil-images/mine/3qnv) | Carboxypeptidase T | Descriptor: | Carboxypeptidase T, GLYCEROL, SULFATE ION, ... | Authors: | Timofeev, V.I, Akparov, V.K, Kuranova, I.P. | Deposit date: | 2011-02-09 | Release date: | 2012-02-15 | Method: | X-RAY DIFFRACTION (1.69 Å) | Cite: | Three-dimensional structure of recombinant carboxypeptidase T from Thermoactinomyces vulgaris without calcium ions Crystallography Reports, 56, 2011
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5MRV
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![BU of 5mrv by Molmil](/molmil-images/mine/5mrv) | Crystal structure of human carboxypeptidase O in complex with NvCI | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Carboxypeptidase O, Metallocarboxypeptidase inhibitor, ... | Authors: | Garcia-Pardo, J, Garcia-Guerrero, M.C, Fernandez-Alvarez, R, Lyons, P, Aviles, F.X, Lorenzo, J, Reverter, D. | Deposit date: | 2016-12-27 | Release date: | 2018-01-17 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.854 Å) | Cite: | Crystal structure and mechanism of human carboxypeptidase O: Insights into its specific activity for acidic residues. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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6SN6
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![BU of 6sn6 by Molmil](/molmil-images/mine/6sn6) | |
5LYF
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![BU of 5lyf by Molmil](/molmil-images/mine/5lyf) | Crystal structure of 1 in complex with tafCPB | Descriptor: | (2~{S})-6-azanyl-2-[[(2~{R})-1-[[(1~{R},2~{S},4~{S})-2-bicyclo[2.2.1]heptanyl]amino]-3-cyclohexyl-1-oxidanylidene-propan-2-yl]carbamoylamino]hexanoic acid, Carboxypeptidase B, ZINC ION | Authors: | Schreuder, H, Liesum, A, Loenze, P. | Deposit date: | 2016-09-28 | Release date: | 2016-10-26 | Last modified: | 2016-12-21 | Method: | X-RAY DIFFRACTION (2.01 Å) | Cite: | Sulfamide as Zinc Binding Motif in Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (TAFIa). J. Med. Chem., 59, 2016
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6T9Y
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![BU of 6t9y by Molmil](/molmil-images/mine/6t9y) | |