6GJD
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![BU of 6gjd by Molmil](/molmil-images/mine/6gjd) | Erk2 signalling protein | Descriptor: | DIMETHYL SULFOXIDE, GLYCEROL, Mitogen-activated protein kinase 1, ... | Authors: | O'Reilly, M. | Deposit date: | 2018-05-16 | Release date: | 2019-01-02 | Method: | X-RAY DIFFRACTION (1.58 Å) | Cite: | Quantitation of ERK1/2 inhibitor cellular target occupancies with a reversible slow off-rate probe. Chem Sci, 9, 2018
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6GJB
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![BU of 6gjb by Molmil](/molmil-images/mine/6gjb) | Erk2 signalling protein | Descriptor: | Mitogen-activated protein kinase 1, SULFATE ION, [(1~{R},4~{Z})-cyclooct-4-en-1-yl] ~{N}-[4-[4-[[4-[1-[(1~{S})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Authors: | O'Reilly, M. | Deposit date: | 2018-05-16 | Release date: | 2019-01-02 | Method: | X-RAY DIFFRACTION (1.82 Å) | Cite: | Quantitation of ERK1/2 inhibitor cellular target occupancies with a reversible slow off-rate probe. Chem Sci, 9, 2018
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6GES
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![BU of 6ges by Molmil](/molmil-images/mine/6ges) | Crystal structure of ERK1 covalently bound to SM1-71 | Descriptor: | 1,2-ETHANEDIOL, Mitogen-activated protein kinase 3, N-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide, ... | Authors: | Chaikuad, A, Suman, R, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Gray, N.S, Knapp, S, Structural Genomics Consortium (SGC) | Deposit date: | 2018-04-27 | Release date: | 2019-02-27 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (2.07 Å) | Cite: | Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome. Cell Chem Biol, 26, 2019
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6GE0
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![BU of 6ge0 by Molmil](/molmil-images/mine/6ge0) | |
6GDQ
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![BU of 6gdq by Molmil](/molmil-images/mine/6gdq) | |
6GDM
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![BU of 6gdm by Molmil](/molmil-images/mine/6gdm) | |
6G9N
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![BU of 6g9n by Molmil](/molmil-images/mine/6g9n) | |
6G9M
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![BU of 6g9m by Molmil](/molmil-images/mine/6g9m) | |
6G9K
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![BU of 6g9k by Molmil](/molmil-images/mine/6g9k) | |
6G9J
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![BU of 6g9j by Molmil](/molmil-images/mine/6g9j) | |
6G9H
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![BU of 6g9h by Molmil](/molmil-images/mine/6g9h) | |
6G9D
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![BU of 6g9d by Molmil](/molmil-images/mine/6g9d) | |
6G9A
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![BU of 6g9a by Molmil](/molmil-images/mine/6g9a) | |
6G97
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![BU of 6g97 by Molmil](/molmil-images/mine/6g97) | |
6G93
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![BU of 6g93 by Molmil](/molmil-images/mine/6g93) | |
6G92
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![BU of 6g92 by Molmil](/molmil-images/mine/6g92) | |
6G91
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![BU of 6g91 by Molmil](/molmil-images/mine/6g91) | |
6G8X
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![BU of 6g8x by Molmil](/molmil-images/mine/6g8x) | |
6G54
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![BU of 6g54 by Molmil](/molmil-images/mine/6g54) | Crystal structure of ERK2 covalently bound to SM1-71 | Descriptor: | 1,2-ETHANEDIOL, CHLORIDE ION, Mitogen-activated protein kinase 1, ... | Authors: | Chaikuad, A, Suman, R, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Gray, N.S, Knapp, S, Structural Genomics Consortium (SGC) | Deposit date: | 2018-03-29 | Release date: | 2019-02-27 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome. Cell Chem Biol, 26, 2019
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6FXV
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![BU of 6fxv by Molmil](/molmil-images/mine/6fxv) | |
6FRP
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![BU of 6frp by Molmil](/molmil-images/mine/6frp) | |
6FR1
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![BU of 6fr1 by Molmil](/molmil-images/mine/6fr1) | |
6FQ7
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![BU of 6fq7 by Molmil](/molmil-images/mine/6fq7) | Crystal structure of ERK2 in complex with an adenosine derivative | Descriptor: | 4-[6-azanyl-9-[(2~{R},3~{R},4~{S},5~{R})-5-(azidomethyl)-3,4-bis(oxidanyl)oxolan-2-yl]purin-8-yl]sulfanylbutanoic acid, DIMETHYL SULFOXIDE, Mitogen-activated protein kinase 1, ... | Authors: | Gelin, M, Labesse, G. | Deposit date: | 2018-02-13 | Release date: | 2019-03-13 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | None To be published
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6FN5
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![BU of 6fn5 by Molmil](/molmil-images/mine/6fn5) | |
6FMA
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![BU of 6fma by Molmil](/molmil-images/mine/6fma) | Crystal structure of ERK2 in complex with an adenosine derivative | Descriptor: | 3-[6-azanyl-9-[(2~{R},3~{R},4~{S},5~{R})-5-(azidomethyl)-3,4-bis(oxidanyl)oxolan-2-yl]purin-8-yl]sulfanylpropanoic acid, DIMETHYL SULFOXIDE, Mitogen-activated protein kinase 1, ... | Authors: | Gelin, M, Labesse, G. | Deposit date: | 2018-01-30 | Release date: | 2019-03-13 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.667 Å) | Cite: | None To be published
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