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1A0M
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1.1 ANGSTROM CRYSTAL STRUCTURE OF A-CONOTOXIN [TYR15]-EPI
分子名称: ALPHA-CONOTOXIN [TYR15]-EPI
著者Hu, S.-H, Loughnan, M, Miller, R, Weeks, C.M, Blessing, R.H, Alewood, P.F, Lewis, R.J, Martin, J.L.
登録日1997-12-03
公開日1999-01-13
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献The 1.1 A resolution crystal structure of [Tyr15]EpI, a novel alpha-conotoxin from Conus episcopatus, solved by direct methods.
Biochemistry, 37, 1998
1AKG
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ALPHA-CONOTOXIN PNIB FROM CONUS PENNACEUS
分子名称: ALPHA-CONOTOXIN PNIB
著者Hu, S.-H, Martin, J.L.
登録日1997-05-18
公開日1998-05-20
最終更新日2015-06-10
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Crystal structure at 1.1 A resolution of alpha-conotoxin PnIB: comparison with alpha-conotoxins PnIA and GI.
Biochemistry, 36, 1997
4TTL
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Racemic structure of cyclic Vc1.1 (cVc1.1-1)
分子名称: Alpha-conotoxin Vc1A
著者Wang, C.K, King, G.J, Craik, D.J.
登録日2014-06-22
公開日2014-09-10
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.7004 Å)
主引用文献Racemic and Quasi-Racemic X-ray Structures of Cyclic Disulfide-Rich Peptide Drug Scaffolds.
Angew.Chem.Int.Ed.Engl., 53, 2014
5CO5
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Crystal structure of Ac-AChBP in complex with conotoxin GIC
分子名称: Alpha-conotoxin GIC, Soluble acetylcholine receptor
著者Wang, X.Q, Xu, M.Y, Luo, S.L, Lin, B.
登録日2015-07-19
公開日2016-07-20
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of Ac-AChBP in complex with conotoxin GIC
To Be Published
5JME
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Crystal structure of acetylcholine binding protein (AChBP) from Aplysia Californica in complex with alpha-conotoxin PeIA
分子名称: Soluble acetylcholine receptor, alpha-conotoxin PeIA from Conus pergrandis
著者Bobango, J, Sankaran, B, McIntosh, J.M, Talley, T.T.
登録日2016-04-28
公開日2016-05-11
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.336 Å)
主引用文献Crystal structure of acetylcholine binding protein (AChBP) from Aplysia Californica in complex with alpha-conotoxin PeIA
To Be Published
7N43
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Alpha-conotoxin OmIA with unusual pharmacological properties at alpha7 nicotinic receptors
分子名称: Acetylcholine-binding protein, Alpha-conotoxin OmIA
著者Ho, T.N.T, Abraham, N, Lewis, R.J.
登録日2021-06-03
公開日2021-12-01
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.47 Å)
主引用文献Unique Pharmacological Properties of alpha-Conotoxin OmIA at alpha 7 nAChRs.
Front Pharmacol, 12, 2021
6M4Z
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Co-crystal structure of Ac-AChBPP in complex with alpha-conotoxin [D11A]LvIA
分子名称: Alpha-conotoxin LvIA, Soluble acetylcholine receptor
著者Wang, X.Q, Pan, S, Luo, S.L, Zhu, X.P.
登録日2020-03-09
公開日2021-03-10
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.803 Å)
主引用文献The crystal structure of Ac-AChBP in complex with LvIA analogs reveals the mechanism of its selectivity towards different nAChR subtypes
To Be Published
6M4X
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Co-crystal structure of Ac-AChBPP in complex with [N9A]LvIA
分子名称: Alpha-conotoxin LvIA, Soluble acetylcholine receptor
著者Wang, X.Q, Pan, S, Luo, S.L, Zhu, X.P.
登録日2020-03-09
公開日2021-03-10
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.998 Å)
主引用文献The crystal structure of Ac-AChBP in complex with LvIA analogs reveals the mechanism of its selectivity towards different nAChR subtypes
To Be Published
5XGL
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Co-crystal structure of Ac-AChBPP in complex with alpha-conotoxin LvIA
分子名称: Alpha-conotoxin LvIA, Soluble acetylcholine receptor
著者Wang, X.Q, Xu, M.Y, Luo, S.L, Zhu, X.P.
登録日2017-04-14
公開日2018-06-13
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.439 Å)
主引用文献The crystal structure of Ac-AChBP in complex with alpha-conotoxin LvIA reveals the mechanism of its selectivity towards different nAChR subtypes
Protein Cell, 8, 2017
7N0T
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NMR structure of EpI[Y(SO)315Y]-OH
分子名称: Alpha-conotoxin EpI
著者Conibear, A.C, Rosengren, K.J, Lee, H.S.
登録日2021-05-26
公開日2021-11-10
最終更新日2024-10-16
実験手法SOLUTION NMR
主引用文献Posttranslational modifications of alpha-conotoxins: sulfotyrosine and C-terminal amidation stabilise structures and increase acetylcholine receptor binding.
Rsc Med Chem, 12, 2021
2M3I
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Characterization of a Novel Alpha4/6-Conotoxin TxIC from Conus textile that Potently Blocks alpha3beta4 Nicotinic Acetylcholine Receptors
分子名称: Alpha-conotoxin
著者Luo, S, Zhangsun, D, Zhu, X, Wu, Y, Hu, Y, Christensen, S, Akcan, M, Craik, D.J, McIntosh, J.M.
登録日2013-01-20
公開日2013-12-04
最終更新日2024-10-16
実験手法SOLUTION NMR
主引用文献Characterization of a Novel alpha-Conotoxin TxID from Conus textile That Potently Blocks Rat alpha 3 beta 4 Nicotinic Acetylcholine Receptors.
J.Med.Chem., 56, 2013
2LZ5
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Solution structure of a Novel Alpha-Conotoxin TxIB
分子名称: Conotoxin_TxIB
著者Luo, S, Zhangsun, D, Wu, Y, Zhu, X, Hu, Y, McIntyre, M, Christensen, S, Akcan, M, Craik, D, McIntosh, J.
登録日2012-09-23
公開日2012-12-05
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Characterization of a novel alpha-conotoxin from conus textile that selectively targets alpha6/alpha3beta2beta3 nicotinic acetylcholine receptors.
J.Biol.Chem., 288, 2013
9BAF
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Solution NMR structure of conofurin-Delta
分子名称: Alpha-conotoxin LvIA
著者Harvey, P.J, Craik, D.J, Hone, A.J, McIntosh, J.M.
登録日2024-04-04
公開日2024-07-03
最終更新日2024-10-16
実験手法SOLUTION NMR
主引用文献Design, Synthesis, and Structure-Activity Relationships of Novel Peptide Derivatives of the Severe Acute Respiratory Syndrome-Coronavirus-2 Spike-Protein that Potently Inhibit Nicotinic Acetylcholine Receptors.
J.Med.Chem., 67, 2024
2MD6
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NMR SOLUTION STRUCTURE OF ALPHA CONOTOXIN LO1A FROM Conus longurionis
分子名称: ALPHA CONOTOXIN LO1A
著者Maiti, M, Lescrinier, E, Herdewijn, P, Lebbe, E.K.M, Peigneur, S, D'Souza, L, Tytgat, J.
登録日2013-09-01
公開日2014-03-05
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structure-Function Elucidation of a New alpha-Conotoxin, Lo1a, from Conus longurionis.
J.Biol.Chem., 289, 2014
7KNN
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Solution structure of the alpha-conotoxin analogue [2-8]-alkyne Vc1.1
分子名称: Alpha-conotoxin Vc1a
著者MacRaild, C.A, Robinson, S.D, Chhabra, S, Norton, R.S.
登録日2020-11-05
公開日2021-09-15
最終更新日2023-11-15
実験手法SOLUTION NMR
主引用文献Alkyne-Bridged alpha-Conotoxin Vc1.1 Potently Reverses Mechanical Allodynia in Neuropathic Pain Models.
J.Med.Chem., 64, 2021
2NAY
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BU of 2nay by Molmil
The structure of the Bt1.8 peptide synthesized by solid-phase method
分子名称: Conotoxin Bt1.8
著者Chenyun, G, Biling, H.
登録日2016-01-14
公開日2016-02-03
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献The structure of the Bt1.8 peptide synthesized by solid-phase method
To be Published
2N07
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Design of a Highly Stable Disulfide-Deleted Mutant of Analgesic Cyclic alpha-Conotoxin Vc1.1
分子名称: Alpha-conotoxin Vc1A
著者Yu, R, Seymour, V, Berecki, G, Jia, X, Akcan, M, Adams, D, Kaas, Q, Craik, D.
登録日2015-03-04
公開日2016-04-13
実験手法SOLUTION NMR
主引用文献Design of a Highly Stable Disulfide-Deleted Mutant of Analgesic Cyclic alpha-Conotoxin Vc1.1.
To be Published
1P1P
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[PRO7,13] AA-CONOTOXIN PIVA, NMR, 12 STRUCTURES
分子名称: AA-CONOTOXIN PIVA
著者Han, K.-H, Hwang, K.-J, Kim, S.-M, Kim, S.-K, Gray, W.R, Olivera, B.M, Rivier, J, Shon, K.J.
登録日1996-12-06
公開日1997-07-07
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献NMR structure determination of a novel conotoxin, [Pro 7,13] alpha A-conotoxin PIVA.
Biochemistry, 36, 1997
2H8S
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Solution structure of alpha-conotoxin Vc1.1
分子名称: Alpha-conotoxin Vc1A
著者Clark, R.J, Fischer, H, Nevin, S.T, Adams, D.J, Craik, D.J.
登録日2006-06-07
公開日2006-06-27
最終更新日2024-10-09
実験手法SOLUTION NMR
主引用文献The Synthesis, Structural Characterization, and Receptor Specificity of the {alpha}-Conotoxin Vc1.1.
J.Biol.Chem., 281, 2006
1UL2
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Solution Conformation of alpha-Conotoxin GIC
分子名称: alpha-conotoxin GIC
著者Chi, S.-W, Kim, D.-H, Olivera, B.M, McIntosh, J.M, Han, K.-H.
登録日2003-09-06
公開日2004-07-20
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Solution conformation of alpha-conotoxin GIC, a novel potent antagonist of alpha3beta2 nicotinic acetylcholine receptors
Biochem.J., 380, 2004
1DG2
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SOLUTION CONFORMATION OF A-CONOTOXIN AUIB
分子名称: A-CONOTOXIN AUIB
著者Cho, J.-H, Mok, K.H, Olivera, B.M, McIntosh, J.M, Park, K.-H, Han, K.-H.
登録日1999-11-23
公開日2000-02-25
最終更新日2022-02-16
実験手法SOLUTION NMR
主引用文献Nuclear magnetic resonance solution conformation of alpha-conotoxin AuIB, an alpha(3)beta(4) subtype-selective neuronal nicotinic acetylcholine receptor antagonist.
J.Biol.Chem., 275, 2000
1ZLC
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Solution Conformation of alpha-conotoxin PIA
分子名称: Alpha-conotoxin PIA
著者Chi, S.-W, Lee, S.-H, Kim, D.-H, Kim, J.-S, Olivera, B.M, McIntosh, J.M, Han, K.-H.
登録日2005-05-05
公開日2006-05-02
最終更新日2022-03-02
実験手法SOLUTION NMR
主引用文献Solution structure of alpha-conotoxin PIA, a novel antagonist of alpha6 subunit containing nicotinic acetylcholine receptors
Biochem.Biophys.Res.Commun., 338, 2005
5UG3
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NMR SOLUTION STRUCTURE OF ALPHA-CONOTOXIN GID MUTANT A10V
分子名称: Alpha-conotoxin GID
著者Hussein, A.K, Leffler, A.E, Zebroski, H.A, Powell, S.R, Kuryatov, A, Filipenko, P, Gorson, J, Heizmann, A, Lyskov, S, Nicke, A, Lindstrom, J, Rudy, B, Bonneau, R, Holford, M, Poget, S.F.
登録日2017-01-06
公開日2017-09-06
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Discovery of peptide ligands through docking and virtual screening at nicotinic acetylcholine receptor homology models.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
5UG5
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NMR SOLUTION STRUCTURE OF THE ALPHA-CONOTOXIN GID MUTANT V13Y
分子名称: Alpha-conotoxin GID
著者Hussein, A, Leffler, A.E, Kuryatov, A, Zebroski, H.A, Powell, S.R, Filipenko, P, Gorson, J, Heizmann, A, Lyskov, S, Nicke, A, Lindstrom, J, Rudy, B, Bonneau, R, Holford, M, Poget, S.F.
登録日2017-01-06
公開日2017-09-06
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Discovery of peptide ligands through docking and virtual screening at nicotinic acetylcholine receptor homology models.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
6OTA
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THREE-DIMENSIONAL STRUCTURE IN SOLUTION OF THE RIBBON DISULFIDE ISOMER OF THE NICOTINIC ACETYLCHOLINE RECEPTOR ANTAGONIST ALPHA-CONOTOXIN TxIA
分子名称: Alpha-conotoxin TxIA
著者Clark, R.J, Nicke, A.
登録日2019-05-02
公開日2020-05-06
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Structural and functional analysis of E. Coli-expressed 4/7 alpha-conotoxin analogues reveals preferential formation of ribbon isomers
To Be Published

 

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